ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development最新文献

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First potent macrocyclic A3adenosine receptor agonists reveal G-protein and beta-arrestin2 signaling preferences 第一种有效的大环腺苷受体激动剂揭示了g蛋白和β -arrestin2信号传导偏好
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.148340
K. Jacobson, Courtney L Fisher, V. Salmaso, Tina C. Wan, Ryan G. Campbell, Eric Chen, Zhang-Guo Gao, J. Auchampach, D. Tosh
{"title":"First potent macrocyclic A3adenosine receptor agonists reveal G-protein and beta-arrestin2 signaling preferences","authors":"K. Jacobson, Courtney L Fisher, V. Salmaso, Tina C. Wan, Ryan G. Campbell, Eric Chen, Zhang-Guo Gao, J. Auchampach, D. Tosh","doi":"10.1124/jpet.122.148340","DOIUrl":"https://doi.org/10.1124/jpet.122.148340","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"1 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"116528149","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Characterization of OJT008 As a Novel Inhibitor ofMycobacterium tuberculosis 新型结核分枝杆菌抑制剂OJT008的研究
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.265640
K. Idowu, Collins Onyenaka, Ngan P. Ha, E. Graviss, Omonike A. Olaleye
{"title":"Characterization of OJT008 As a Novel Inhibitor ofMycobacterium tuberculosis","authors":"K. Idowu, Collins Onyenaka, Ngan P. Ha, E. Graviss, Omonike A. Olaleye","doi":"10.1124/jpet.122.265640","DOIUrl":"https://doi.org/10.1124/jpet.122.265640","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"25 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"134455005","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Development of highly potent and selective inhibitors for GRK5 高效选择性GRK5抑制剂的开发
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.140620
Yueyi Chen
{"title":"Development of highly potent and selective inhibitors for GRK5","authors":"Yueyi Chen","doi":"10.1124/jpet.122.140620","DOIUrl":"https://doi.org/10.1124/jpet.122.140620","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"522 ","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"113997370","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Phytochemotypic profiling and GCMS Analysis ofViola patrinii, a Himalayan Herb 喜马拉雅草本植物堇菜的植物化学型分析及GCMS分析
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.242400
Sajad Yousuf, Tahir Yousuf, O. Morenikeji, Naseer A Kutchy
{"title":"Phytochemotypic profiling and GCMS Analysis ofViola patrinii, a Himalayan Herb","authors":"Sajad Yousuf, Tahir Yousuf, O. Morenikeji, Naseer A Kutchy","doi":"10.1124/jpet.122.242400","DOIUrl":"https://doi.org/10.1124/jpet.122.242400","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"33 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123844515","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Sildenafil is a candidate drug for Alzheimer's disease: Real-world patient and RNA-sequencing data observations in patient-induced pluripotent stem cells-derived neurons 西地那非是阿尔茨海默病的候选药物:现实世界患者和患者诱导的多能干细胞来源神经元的rna测序数据观察
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.526220
Yichen Li, D. Gohel, Pengyue Zhang, Chienwei Chiang, A. Pieper, J. Cummings, F. Cheng
{"title":"Sildenafil is a candidate drug for Alzheimer's disease: Real-world patient and RNA-sequencing data observations in patient-induced pluripotent stem cells-derived neurons","authors":"Yichen Li, D. Gohel, Pengyue Zhang, Chienwei Chiang, A. Pieper, J. Cummings, F. Cheng","doi":"10.1124/jpet.122.526220","DOIUrl":"https://doi.org/10.1124/jpet.122.526220","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"35 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"122329078","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Design, Synthesis and Biological Evaluation of Benzothiazole-Phenyl Analogs as Multi-Target Directed Ligands for Treating Pain 苯并噻唑-苯基类似物多靶点定向配体治疗疼痛的设计、合成和生物学评价
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.143050
S. Pecic, Jeannes Angelia, Xiaohui Weng
{"title":"Design, Synthesis and Biological Evaluation of Benzothiazole-Phenyl Analogs as Multi-Target Directed Ligands for Treating Pain","authors":"S. Pecic, Jeannes Angelia, Xiaohui Weng","doi":"10.1124/jpet.122.143050","DOIUrl":"https://doi.org/10.1124/jpet.122.143050","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"258 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123966977","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Analgesic and Side Effect Profiles of Novel Alpha-2 Adrenergic Receptor Agonists 新型α -2肾上腺素能受体激动剂的镇痛和副作用
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.241500
Cristina D. Peterson, Lukas D. Caye, K. Kitto, G. Wilcox, Laura S. Stone, Swati More, C. Fairbanks
{"title":"Analgesic and Side Effect Profiles of Novel Alpha-2 Adrenergic Receptor Agonists","authors":"Cristina D. Peterson, Lukas D. Caye, K. Kitto, G. Wilcox, Laura S. Stone, Swati More, C. Fairbanks","doi":"10.1124/jpet.122.241500","DOIUrl":"https://doi.org/10.1124/jpet.122.241500","url":null,"abstract":",","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"128 3 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"129973067","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
In vitroantiglycation and protein cross-link breakage effects ofMurraya koenigiileaf extracts and their phytochemical composition 木参提取物的体外抗糖化和蛋白质交联断裂作用及其植物化学成分
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.286220
O. Adeniran, S. Gololo
{"title":"In vitroantiglycation and protein cross-link breakage effects ofMurraya koenigiileaf extracts and their phytochemical composition","authors":"O. Adeniran, S. Gololo","doi":"10.1124/jpet.122.286220","DOIUrl":"https://doi.org/10.1124/jpet.122.286220","url":null,"abstract":"ID 28622","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"24 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"120960003","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Efficacy of HS-10382 (TERN-701) in tumor xenograft models, a new investigational allosteric ABL1 kinase inhibitor as a potential treatment for CML HS-10382 (TERN-701)在肿瘤异种移植模型中的疗效,一种新的研究变构ABL1激酶抑制剂作为CML的潜在治疗方法
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.533280
Yuanfeng Zhou, Benjamin Parsons, Danni Sun, Yunfan Li, Guoliang Chen, Mingjie Luo, Christopher Jones, Xiaogang Lian, Xiaolei Wang, Yundong Sun, Jeffrey Jasper, H. Niu
{"title":"Efficacy of HS-10382 (TERN-701) in tumor xenograft models, a new investigational allosteric ABL1 kinase inhibitor as a potential treatment for CML","authors":"Yuanfeng Zhou, Benjamin Parsons, Danni Sun, Yunfan Li, Guoliang Chen, Mingjie Luo, Christopher Jones, Xiaogang Lian, Xiaolei Wang, Yundong Sun, Jeffrey Jasper, H. Niu","doi":"10.1124/jpet.122.533280","DOIUrl":"https://doi.org/10.1124/jpet.122.533280","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"517 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123103345","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Novel Axin Stabilizer YA6060 is a Promising Therapy for Liver Fibrosis 新型轴蛋白稳定剂YA6060有望治疗肝纤维化
ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development Pub Date : 2023-05-18 DOI: 10.1124/jpet.122.176280
Yan Shu, Shiwei Zhou, Yong Ai, Shaoteng Wang, A. Xu, F. Xue
{"title":"Novel Axin Stabilizer YA6060 is a Promising Therapy for Liver Fibrosis","authors":"Yan Shu, Shiwei Zhou, Yong Ai, Shaoteng Wang, A. Xu, F. Xue","doi":"10.1124/jpet.122.176280","DOIUrl":"https://doi.org/10.1124/jpet.122.176280","url":null,"abstract":"","PeriodicalId":173142,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Drug Discovery and Development","volume":"26 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131074363","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
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