{"title":"False Resistance to Antiparasitic Drugs: Causes from Shelf Availability to Patient Compliance","authors":"J. Cabaret","doi":"10.2174/1871521411009030161","DOIUrl":"https://doi.org/10.2174/1871521411009030161","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"161-167"},"PeriodicalIF":0.0,"publicationDate":"2010-06-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68024676","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
E. Co, S. Johnson, T. Murthy, M. Talwar, M. Hickman, Jacob D. Johnson
{"title":"Recent Methods in Antimalarial Susceptibility Testing","authors":"E. Co, S. Johnson, T. Murthy, M. Talwar, M. Hickman, Jacob D. Johnson","doi":"10.2174/1871521411009030148","DOIUrl":"https://doi.org/10.2174/1871521411009030148","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"148-160"},"PeriodicalIF":0.0,"publicationDate":"2010-06-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/1871521411009030148","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68024663","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Recent Development and Future Perspective of Antitubercular Therapy","authors":"M. Chhabria, Shailesh M. Patel, M. Jani","doi":"10.2174/187152110791383779","DOIUrl":"https://doi.org/10.2174/187152110791383779","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"59-103"},"PeriodicalIF":0.0,"publicationDate":"2010-03-31","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023584","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Lactobacillus GG (LGG) Peptides Can Inhibit Antibiotic-Resistant Bacteria Growth","authors":"R. Lu, J. Nataro, A. Fasano","doi":"10.2174/187152110791383760","DOIUrl":"https://doi.org/10.2174/187152110791383760","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"48-51"},"PeriodicalIF":0.0,"publicationDate":"2010-03-31","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152110791383760","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023539","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Chem-Bioinformatics : Computational Modeling of TIBO Derivatives","authors":"A. Thakur, M. Thakur, N. Agrawal, S. Bhadoria","doi":"10.2174/187152110791383751","DOIUrl":"https://doi.org/10.2174/187152110791383751","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"52-58"},"PeriodicalIF":0.0,"publicationDate":"2010-03-31","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023525","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"From Vancomycin to Oritavancin: The Discovery and Development of a Novel Lipoglycopeptide Antibiotic","authors":"N. E. Allen","doi":"10.2174/187152110790886745","DOIUrl":"https://doi.org/10.2174/187152110790886745","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"23-47"},"PeriodicalIF":0.0,"publicationDate":"2010-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152110790886745","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023494","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
K. Brandenburg, J. Howe, S. Sanchez-Gomez, P. Garidel, M. Roessle, J. Andrä, R. Jerala, Dagmar Zweytick, K. Lohner, M. Rappolt, S. Blondelle, I. Moriyón, G. Tejada
{"title":"Effective Antimicrobial and Anti-Endotoxin Activity of Cationic Peptides Based on Lactoferricin: A Biophysical and Microbiological Study","authors":"K. Brandenburg, J. Howe, S. Sanchez-Gomez, P. Garidel, M. Roessle, J. Andrä, R. Jerala, Dagmar Zweytick, K. Lohner, M. Rappolt, S. Blondelle, I. Moriyón, G. Tejada","doi":"10.2174/187152110790886736","DOIUrl":"https://doi.org/10.2174/187152110790886736","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"9-22"},"PeriodicalIF":0.0,"publicationDate":"2010-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152110790886736","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023480","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Small Molecule Approaches Toward the Non-Microbicidal Modulation of Bacterial Biofilm Growth and Maintenance","authors":"Justin J. Richards and Christian Melander","doi":"10.2174/187152109789760135","DOIUrl":"https://doi.org/10.2174/187152109789760135","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"8 1","pages":"295-314"},"PeriodicalIF":0.0,"publicationDate":"2009-09-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023329","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
J. Pollard, Jonathan O. Wright, Yanshu Feng, Dianliang Geng, C. Genberg, P. Savage
{"title":"Activities of Ceragenin CSA-13 Against Established Biofilms in an In Vitro Model of Catheter Decolonization","authors":"J. Pollard, Jonathan O. Wright, Yanshu Feng, Dianliang Geng, C. Genberg, P. Savage","doi":"10.2174/187152109789760225","DOIUrl":"https://doi.org/10.2174/187152109789760225","url":null,"abstract":"Bacterial biofilms on medical devices are a primary source of infection, and efforts have been made to develop means of decontaminating colonized devices including hemodialysis catheter \"lock\" solutions. Because bacterial biofilms are inherently resistant to many antibiotics and widespread use of antibiotics contributes to resistance development, there is a need for new approaches to biofilm eradication. We have developed a class of compounds, termed ceragenins, that mimic the antimicrobial activities of antimicrobial peptides. The ceragenins are active against established biofilms. We tested solutions of a lead ceragenin, CSA-13, with and without EGTA against biofilms comprised of Gram-negative and positive organisms. Similar solutions containing ciprofloxacin were used as comparators. The ceragenin solutions eradi- cated biofilms at concentrations comparable to those required for eradication by ciprofloxacin. However, against a methi- cillin-resistant strain of Staphylococcus aureus, CSA-13 proved to be far superior to ciprofloxacin.","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"8 1","pages":"290-294"},"PeriodicalIF":0.0,"publicationDate":"2009-09-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023456","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Quorum-sensing inhibitors and biofilms","authors":"Martin G. Kociolek","doi":"10.2174/187152109789760117","DOIUrl":"https://doi.org/10.2174/187152109789760117","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"8 1","pages":"315-326"},"PeriodicalIF":0.0,"publicationDate":"2009-09-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152109789760117","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023289","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}