Anti-infective agents in medicinal chemistry最新文献

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False Resistance to Antiparasitic Drugs: Causes from Shelf Availability to Patient Compliance 抗寄生虫药物的虚假耐药性:从货架可用性到患者依从性的原因
Anti-infective agents in medicinal chemistry Pub Date : 2010-06-30 DOI: 10.2174/1871521411009030161
J. Cabaret
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引用次数: 5
Recent Methods in Antimalarial Susceptibility Testing 抗疟药敏试验新方法
Anti-infective agents in medicinal chemistry Pub Date : 2010-06-30 DOI: 10.2174/1871521411009030148
E. Co, S. Johnson, T. Murthy, M. Talwar, M. Hickman, Jacob D. Johnson
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引用次数: 5
Recent Development and Future Perspective of Antitubercular Therapy 抗结核治疗的最新进展及未来展望
Anti-infective agents in medicinal chemistry Pub Date : 2010-03-31 DOI: 10.2174/187152110791383779
M. Chhabria, Shailesh M. Patel, M. Jani
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引用次数: 10
Lactobacillus GG (LGG) Peptides Can Inhibit Antibiotic-Resistant Bacteria Growth 乳酸菌GG (LGG)肽可抑制耐药菌生长
Anti-infective agents in medicinal chemistry Pub Date : 2010-03-31 DOI: 10.2174/187152110791383760
R. Lu, J. Nataro, A. Fasano
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引用次数: 2
Chem-Bioinformatics : Computational Modeling of TIBO Derivatives 化学生物信息学:TIBO衍生物的计算建模
Anti-infective agents in medicinal chemistry Pub Date : 2010-03-31 DOI: 10.2174/187152110791383751
A. Thakur, M. Thakur, N. Agrawal, S. Bhadoria
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引用次数: 1
From Vancomycin to Oritavancin: The Discovery and Development of a Novel Lipoglycopeptide Antibiotic 从万古霉素到奥利塔万辛:一种新型脂糖肽抗生素的发现与发展
Anti-infective agents in medicinal chemistry Pub Date : 2010-01-01 DOI: 10.2174/187152110790886745
N. E. Allen
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引用次数: 34
Effective Antimicrobial and Anti-Endotoxin Activity of Cationic Peptides Based on Lactoferricin: A Biophysical and Microbiological Study 基于乳铁蛋白的阳离子多肽有效抗菌和抗内毒素活性:生物物理和微生物学研究
Anti-infective agents in medicinal chemistry Pub Date : 2010-01-01 DOI: 10.2174/187152110790886736
K. Brandenburg, J. Howe, S. Sanchez-Gomez, P. Garidel, M. Roessle, J. Andrä, R. Jerala, Dagmar Zweytick, K. Lohner, M. Rappolt, S. Blondelle, I. Moriyón, G. Tejada
{"title":"Effective Antimicrobial and Anti-Endotoxin Activity of Cationic Peptides Based on Lactoferricin: A Biophysical and Microbiological Study","authors":"K. Brandenburg, J. Howe, S. Sanchez-Gomez, P. Garidel, M. Roessle, J. Andrä, R. Jerala, Dagmar Zweytick, K. Lohner, M. Rappolt, S. Blondelle, I. Moriyón, G. Tejada","doi":"10.2174/187152110790886736","DOIUrl":"https://doi.org/10.2174/187152110790886736","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"9 1","pages":"9-22"},"PeriodicalIF":0.0,"publicationDate":"2010-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152110790886736","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023480","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 10
Small Molecule Approaches Toward the Non-Microbicidal Modulation of Bacterial Biofilm Growth and Maintenance 非杀微生物调控细菌生物膜生长和维持的小分子方法
Anti-infective agents in medicinal chemistry Pub Date : 2009-09-30 DOI: 10.2174/187152109789760135
Justin J. Richards and Christian Melander
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引用次数: 27
Activities of Ceragenin CSA-13 Against Established Biofilms in an In Vitro Model of Catheter Decolonization Ceragenin CSA-13在导管离体模型中对已建立生物膜的活性研究
Anti-infective agents in medicinal chemistry Pub Date : 2009-09-30 DOI: 10.2174/187152109789760225
J. Pollard, Jonathan O. Wright, Yanshu Feng, Dianliang Geng, C. Genberg, P. Savage
{"title":"Activities of Ceragenin CSA-13 Against Established Biofilms in an In Vitro Model of Catheter Decolonization","authors":"J. Pollard, Jonathan O. Wright, Yanshu Feng, Dianliang Geng, C. Genberg, P. Savage","doi":"10.2174/187152109789760225","DOIUrl":"https://doi.org/10.2174/187152109789760225","url":null,"abstract":"Bacterial biofilms on medical devices are a primary source of infection, and efforts have been made to develop means of decontaminating colonized devices including hemodialysis catheter \"lock\" solutions. Because bacterial biofilms are inherently resistant to many antibiotics and widespread use of antibiotics contributes to resistance development, there is a need for new approaches to biofilm eradication. We have developed a class of compounds, termed ceragenins, that mimic the antimicrobial activities of antimicrobial peptides. The ceragenins are active against established biofilms. We tested solutions of a lead ceragenin, CSA-13, with and without EGTA against biofilms comprised of Gram-negative and positive organisms. Similar solutions containing ciprofloxacin were used as comparators. The ceragenin solutions eradi- cated biofilms at concentrations comparable to those required for eradication by ciprofloxacin. However, against a methi- cillin-resistant strain of Staphylococcus aureus, CSA-13 proved to be far superior to ciprofloxacin.","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"8 1","pages":"290-294"},"PeriodicalIF":0.0,"publicationDate":"2009-09-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023456","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 18
Quorum-sensing inhibitors and biofilms 群体感应抑制剂和生物膜
Anti-infective agents in medicinal chemistry Pub Date : 2009-09-30 DOI: 10.2174/187152109789760117
Martin G. Kociolek
{"title":"Quorum-sensing inhibitors and biofilms","authors":"Martin G. Kociolek","doi":"10.2174/187152109789760117","DOIUrl":"https://doi.org/10.2174/187152109789760117","url":null,"abstract":"","PeriodicalId":89320,"journal":{"name":"Anti-infective agents in medicinal chemistry","volume":"8 1","pages":"315-326"},"PeriodicalIF":0.0,"publicationDate":"2009-09-30","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.2174/187152109789760117","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"68023289","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 63
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