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Fly Ash:Sulfated Bi2O3-catalyzed Synthesis of Bioactive Arylimines and Arylamines 粉煤灰：硫酸bi2o3催化合成生物活性芳胺和芳胺
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S1070428024110137
S. Nalini, P. Gayathri, J. Divya, I. Muthuvel, K. Thirumurthy, P. Mayavel, N. Dinesh Kumar, G. Thirunarayanan
{"title":"Fly Ash:Sulfated Bi2O3-catalyzed Synthesis of Bioactive Arylimines and Arylamines","authors":"S. Nalini,&nbsp;P. Gayathri,&nbsp;J. Divya,&nbsp;I. Muthuvel,&nbsp;K. Thirumurthy,&nbsp;P. Mayavel,&nbsp;N. Dinesh Kumar,&nbsp;G. Thirunarayanan","doi":"10.1134/S1070428024110137","DOIUrl":"10.1134/S1070428024110137","url":null,"abstract":"<p>Series of arylimines and arylamines were synthesized by the fly ash:sulfated Bi<sub>2</sub>O<sub>3</sub><b>-</b>catalyzed condensations of amines and aldehydes or 3-aminocarbazole and aryl enones under MW irradiation in solvent-free conditions in yields of higher than 60%. The synthesized compounds were characterized by their physical constants and spectroscopic data. The XRD structure of one of the synthesized imines, specifically (<i>E</i>)-<i>N</i>-(2,5-dimethoxybenzylidene)-2-phenoxyaniline imine was obtained. A molecular docking study of the synthesized arylimines and arylamines was performed, and their antimicrobial and antimalarial activities were assessed.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2242 - 2258"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143109285","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Approaches to the Formation of the Key 2-Oxabicyclo[3.3.0]octan-3-one Precursor of Galiellalactone 盖利内酯关键2-氧沙比环[3.3.0]辛烷-3- 1前体的形成途径
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S107042802411006X
A. M. Gimazetdinov, V. V. Zagitov, Z. R. Makaev
{"title":"Approaches to the Formation of the Key 2-Oxabicyclo[3.3.0]octan-3-one Precursor of Galiellalactone","authors":"A. M. Gimazetdinov,&nbsp;V. V. Zagitov,&nbsp;Z. R. Makaev","doi":"10.1134/S107042802411006X","DOIUrl":"10.1134/S107042802411006X","url":null,"abstract":"<p>New vicinal all-<i>cis</i>-trisubstituted derivatives of cyclopentane- and cyclopentenetriols were synthesized.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2130 - 2139"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://link.springer.com/content/pdf/10.1134/S107042802411006X.pdf","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143107899","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"OA","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Three-Component Synthesis of Novel 5H-[1,3]dioxolo[4,5-f]indole Derivatives 新型5H-[1,3]二恶唑[4,5-f]吲哚衍生物的三组分合成
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S1070428024110174
Dan-Dan Wan, Ji Li, Jia-Yan Liu, Dong-Sheng Chen
{"title":"Three-Component Synthesis of Novel 5H-[1,3]dioxolo[4,5-f]indole Derivatives","authors":"Dan-Dan Wan,&nbsp;Ji Li,&nbsp;Jia-Yan Liu,&nbsp;Dong-Sheng Chen","doi":"10.1134/S1070428024110174","DOIUrl":"10.1134/S1070428024110174","url":null,"abstract":"<p>New 5<i>H</i>-[1,3]dioxolo[4,5-<i>f</i>]indole derivatives were synthesized in good yields were synthesized by a one-pot, three-component reaction of benzo[<i>d</i>][1,3]dioxol-5-amine, arylglyoxals, and 4-hydroxyquinolin-2(1<i>H</i>)-one in the presence of acetic acid as a catalyst in an ethanol medium under reflux.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2290 - 2297"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143109680","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Design, Synthesis, and Antibacterial Activity of Morpholine-4-sulfonamide Derivatives morpholin -4-磺酰胺衍生物的设计、合成及抗菌活性研究
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S1070428024110149
Huimin Zou, Yi Tan, Zhiyou Huang, Ping Yang, Wenxia Ou, Xiaohong Li
{"title":"Design, Synthesis, and Antibacterial Activity of Morpholine-4-sulfonamide Derivatives","authors":"Huimin Zou,&nbsp;Yi Tan,&nbsp;Zhiyou Huang,&nbsp;Ping Yang,&nbsp;Wenxia Ou,&nbsp;Xiaohong Li","doi":"10.1134/S1070428024110149","DOIUrl":"10.1134/S1070428024110149","url":null,"abstract":"<p>In the search for novel antibacterial agents, a series of <i>N</i>-(substituted nitrophenyl)morpholine-4-sulfonamides were prepared by the reactions of substituted nitrobenzenes with morpholine-4-sulfonamide under MW irradiation. The synthetic approach is characterized by a facile procedure and broad substrate scope. Preliminary biological assessment of the activity of compounds <b>1b–1h</b>, <b>1k–1n</b> against <i>Xanthomonas oryzae</i> pv. <i>oryzae</i> (<i>Xoo</i>) was higher than 80% at 800 μg/mL. Especially, the inhibition rate of compounds <b>1d</b>, <b>1k</b>, and <b>1n</b> were higher than 95%. Significantly, the EC<sub>50</sub> value of <b>1d</b> was close to the sanguinarine.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2259 - 2265"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143109409","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Electrochemical Carboxylation with CO2 (A Review) 电化学CO2羧化反应（综述）
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S1070428024110010
Yu. H. Budnikova
{"title":"Electrochemical Carboxylation with CO2 (A Review)","authors":"Yu. H. Budnikova","doi":"10.1134/S1070428024110010","DOIUrl":"10.1134/S1070428024110010","url":null,"abstract":"<p>Carbon dioxide (CO<sub>2</sub>) is a widespread, inexpensive, and renewable source of C1 carbon and the main component of greenhouse gases. Therefore, studies on its efficient conversion into useful products, corresponding to the principles of sustainable development, have received considerable attention in recent years. Electrochemical organic synthesis, as an environmentally friendly, mild, and selective approach, is considered an ideal tool for the utilization of CO<sub>2</sub> and its use as a reagent. This review summarizes recent advances in the field of electrocarboxylation involving CO<sub>2</sub> as a precursor in reactions of various types, which reveal a high potential of such transformations in the synthesis of green organics. Special attention is given to processes at the late stage of functionalization of complex molecules that are promising for use in pharmaceutical chemistry.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2055 - 2085"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143109611","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Recent Advances in (Di)Azafluorene Chemistry (A Review) （二）氮杂芴化学进展（综述）
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-27 DOI: 10.1134/S1070428024110022
E. B. Rakhimova, V. Yu. Kirsanov
{"title":"Recent Advances in (Di)Azafluorene Chemistry (A Review)","authors":"E. B. Rakhimova,&nbsp;V. Yu. Kirsanov","doi":"10.1134/S1070428024110022","DOIUrl":"10.1134/S1070428024110022","url":null,"abstract":"<p>The review systematizes and summarizes recent results on the synthesis of aza- and diazafluorenes and their physicochemical properties and biological activity.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 11","pages":"2086 - 2107"},"PeriodicalIF":0.8,"publicationDate":"2025-01-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"143109612","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Green Synthesis of Bioactive Polyhydroquinoline Derivatives via Hantzsch Condensation Using Sulfanilic Acid as a Versatile and Efficient Catalyst 以磺胺酸为高效催化剂，Hantzsch缩合法绿色合成生物活性聚对苯二酚衍生物
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-11 DOI: 10.1134/S1070428024130165
Manoj P. Palve, Jaysing M. Dinore, Amol V. Sapkal, Ajeet A. Yelwande, Rajita D. Ingle
{"title":"Green Synthesis of Bioactive Polyhydroquinoline Derivatives via Hantzsch Condensation Using Sulfanilic Acid as a Versatile and Efficient Catalyst","authors":"Manoj P. Palve,&nbsp;Jaysing M. Dinore,&nbsp;Amol V. Sapkal,&nbsp;Ajeet A. Yelwande,&nbsp;Rajita D. Ingle","doi":"10.1134/S1070428024130165","DOIUrl":"10.1134/S1070428024130165","url":null,"abstract":"<p>A straightforward and efficient synthetic approach for creating polyhydroquinoline derivatives by the Hantzsch reaction using sulfanilic acid as a versatile and efficient catalyst has been proposed. These polyhydroquinoline derivatives are notable for their diverse forms of biological activity. The structures of the synthesized compounds were confirmed using spectroscopic techniques. This methodology provides several advantages, including high yields, cost-effectiveness, time efficiency, environmental friendliness, and operational simplicity.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 1 supplement","pages":"S121 - S127"},"PeriodicalIF":0.8,"publicationDate":"2025-01-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"142940946","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis, Biological Activity, and Molecular Docking Study of New Triazoline Derivatives Using 2-Amino-5-p-subtituted Phenyl-1,3,4-thiadiazoles 2-氨基-5-对取代苯基-1,3,4-噻二唑类新型三唑啉衍生物的合成、生物活性及分子对接研究
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-11 DOI: 10.1134/S1070428024130104
Khadija Najah Zaidane, Ahmed Wahed Naser
{"title":"Synthesis, Biological Activity, and Molecular Docking Study of New Triazoline Derivatives Using 2-Amino-5-p-subtituted Phenyl-1,3,4-thiadiazoles","authors":"Khadija Najah Zaidane,&nbsp;Ahmed Wahed Naser","doi":"10.1134/S1070428024130104","DOIUrl":"10.1134/S1070428024130104","url":null,"abstract":"<p>In this study, new heterocyclic compounds containing 1,3,4-thiadiazole derivatives were synthesized. FT-IR, <sup>1</sup>H NMR, and <sup>13</sup>C NMR spectroscopy were used to identify the title compounds. In addition, some produced compounds were tested <i>in vitro</i> to assess their antimicrobial effectiveness against various microorganisms such as <i>Escherichia coli</i> and <i>Staphylococcus aureus</i>, demonstrating that some of these compounds exhibit very good antibacterial activity. Molecular docking of some of the synthesized compounds showed good results. 1,3,4-Thiadiazole derivatives (<b>1a</b>, <b>1b</b>) were prepared by a reaction of <i>p</i>-nitrobenzoic acid or <i>p</i>-toluic acid with thiosemicarbazide in the presence of POCl<sub>3</sub>. Alkylation of compounds <b>1a</b>,<b> 1b</b> with allyl bromide produced <i>N</i>-allyl thiadiazoles <b>2a</b>, <b>2b</b>. Cyclization of the prepared <i>p</i>-substituted azidobenzene and alkyl azides with compounds <b>2a</b>, <b>2b</b> resulted in the corresponding 1,4-disubstituted triazoline derivatives <b>3a</b>–<b>3h</b> and <b>4a</b>–<b>4d</b>. Molecular docking studies with the target 6ul7 indicated favorable docking scores and binding interactions for the newly synthesized compounds, highlighting their potential as effective antimicrobial agents.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 1 supplement","pages":"S70 - S77"},"PeriodicalIF":0.8,"publicationDate":"2025-01-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"142940954","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Design and Synthesis of Some Novel Phosphorus Heterocycles-Based Coumarin Derivatives as Promising Anticancer Agents 新型磷杂环香豆素类抗癌药物的设计与合成
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-11 DOI: 10.1134/S1070428024130268
N. M. Hassanin, T. E. Ali, M. A. Assiri, S. M. Abdel-Kariem
{"title":"Design and Synthesis of Some Novel Phosphorus Heterocycles-Based Coumarin Derivatives as Promising Anticancer Agents","authors":"N. M. Hassanin,&nbsp;T. E. Ali,&nbsp;M. A. Assiri,&nbsp;S. M. Abdel-Kariem","doi":"10.1134/S1070428024130268","DOIUrl":"10.1134/S1070428024130268","url":null,"abstract":"<p>An efficient method was developed for the synthesis of eight novel functionalized 1,2,4,3-triazaphospholes and one 1,3,2-thiazaphosphinine incorporating a coumarin ring. Additionally, two interesting examples of diethyl coumarinyl phosphonate and diethyl chromeno-[3,4-<i>c</i>][1,2,4]triazolo[4,3-<i>a</i>]pyridinyl phosphonate were obtained. The proposed methodology involved the treatment of <i>N'</i>-benzoyl-2-oxo-2<i>H</i>-chromene-3-carbohydrazonamide (<b>2</b>) with various phosphorus agents, including phosphorus halides, phosphorus triamide, phosphorus esters, and phosphorus sulfides. IR, NMR, and mass spectrometric methods were used to confirm the structures of the prepared compounds. The antiproliferative properties of the isolated compounds were screened against HepG-2, MCF-7, and A549 cancer cells. The products <b>5</b>, <b>7</b>, <b>9</b>, and <b>10</b> exhibited excellent cytotoxic properties compared with doxorubicin. These four bioactive compounds have low toxicity in healthy human HFB4 cells.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 1 supplement","pages":"S223 - S235"},"PeriodicalIF":0.8,"publicationDate":"2025-01-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"142941082","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Solvent-Free Synthesis of Pyrazole Derivatives Mediated by Cobalt-Doped Iron Tartarate 掺杂钴酒石酸铁介导的吡唑衍生物的无溶剂合成
IF 0.8 4区 化学
Russian Journal of Organic Chemistry Pub Date : 2025-01-11 DOI: 10.1134/S1070428024130013
S. B. Jagtap, A. S. Patki, D. B. Muley
{"title":"Solvent-Free Synthesis of Pyrazole Derivatives Mediated by Cobalt-Doped Iron Tartarate","authors":"S. B. Jagtap,&nbsp;A. S. Patki,&nbsp;D. B. Muley","doi":"10.1134/S1070428024130013","DOIUrl":"10.1134/S1070428024130013","url":null,"abstract":"<p>A novel, green, and economically viable method for the one-pot synthesis of 5-amino pyrazole 4-carbonitrile has been established. This approach features the solvent-free reaction between substituted benzaldehyde, malononitrile, and phenyl hydrazine catalyzed by CoFe<sub>2</sub>(C<sub>4</sub>H<sub>4</sub>O<sub>6</sub>)<sub>3</sub>·6H<sub>2</sub>O. The elimination of solvent renders this methodology highly attractive from both cost-effective and environmental perspective. Moreover, the optimized reaction conditions offer operational simplicity, utilize readily available and affordable starting materials, and deliver good to excellent yields (72–92%). The versatility of this protocol is demonstrated by the successful synthesis of ten distinct pyrazole derivatives.</p>","PeriodicalId":766,"journal":{"name":"Russian Journal of Organic Chemistry","volume":"60 1 supplement","pages":"S1 - S8"},"PeriodicalIF":0.8,"publicationDate":"2025-01-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"142941272","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
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