{"title":"Receptor-mediated activation of tyrosine hydroxylase by corticotropin-releasing factor in striatal synaptosomes","authors":"Maria C. Olianas, Pierlugi Onali","doi":"10.1016/S0031-6989(88)80744-6","DOIUrl":"10.1016/S0031-6989(88)80744-6","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1097-1098"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80744-6","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14042080","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
R. Della Loggia , E. Ragazzi , A. Tubaro , G. Fassina , R. Vertua
{"title":"Anti-inflammatory activity of benzopyrones that are inhibitors of cyclo- and lipo-oxygenase","authors":"R. Della Loggia , E. Ragazzi , A. Tubaro , G. Fassina , R. Vertua","doi":"10.1016/S0031-6989(88)80849-X","DOIUrl":"10.1016/S0031-6989(88)80849-X","url":null,"abstract":"<div><p>The anti-inflammatory activity of three benzo-pyrones with prevalent lipooxigenase-inhibitory activity was studied using the Croton oil ear test in mice, in comparison with nordihydroguaieretic acid (NDGA) and indomethacin. Kaempferol, quercetin and NOGA possess a strong and prolonged anti-inflammatory effect, whereas the action of indomethacin appears relevant, but not long-lasting. In contrast the anti-inflammatory activity of esculetin is rather weak, but persistent.</p></div>","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 ","pages":"Pages 91-94"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80849-X","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14280996","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Inhibitory activity of 2-benzimidazolylurea on gastric acid secretion in rats","authors":"S. Trivulzio","doi":"10.1016/S0031-6989(88)80725-2","DOIUrl":"10.1016/S0031-6989(88)80725-2","url":null,"abstract":"<div><p>2-Benzimidazolylurea (BIU) decreases gastric acid secretion. The antisecretive activity appears to be associated with antihistaminic and antimuscarinic effects.</p><p>The antihistaminic activity of BIU appears from its inhibitory effects on betazole stimulated gastric acid secretion and from its inhibitory activity on the isolated guinea pig auricle stimulated by betazole.</p><p>The antimuscarinic activity of BIU appears from several experiments: this molecule decreases gastric acid secretion stimulated by carbachol in rats, depresses the neostigmine-stimulated motility of duodenum in the anaesthetized cat, lessens the hypertonus of isolated guinea pig trachea caused by pylocarpine and also inhibits guinea pig ileum activity stimulated by acetylcholine.</p><p>BIU probably depresses gastric acid secretion by interferring with both histamine and acetylcholine receptors.</p></div>","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1035-1046"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80725-2","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14341170","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"5-HT3 receptors antagonists block morphine- and nicotine- but not amphetamine-induced place-preference conditioning","authors":"E. Acquas, E. Carboni, P. Leone, G. Di Chiara","doi":"10.1016/S0031-6989(88)80752-5","DOIUrl":"10.1016/S0031-6989(88)80752-5","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1113-1114"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80752-5","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14341182","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
E. Landolfi , T. Florio , O. Meucci , M. Grimaldi , G. Magri , D.A. Leong , G. Schettini
{"title":"Steroid modulation of prolactin release from single lactotropes in male and female rats studied by the reverse hemolytic plaque assay","authors":"E. Landolfi , T. Florio , O. Meucci , M. Grimaldi , G. Magri , D.A. Leong , G. Schettini","doi":"10.1016/S0031-6989(88)80733-1","DOIUrl":"10.1016/S0031-6989(88)80733-1","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1075-1076"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80733-1","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14195023","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Caciagli F. , Ciccarelli R. , Di Iorio P. , Traversa U.
{"title":"Autoregulation of endogenous purine release from rat hippocampal slices","authors":"Caciagli F. , Ciccarelli R. , Di Iorio P. , Traversa U.","doi":"10.1016/S0031-6989(88)80731-8","DOIUrl":"10.1016/S0031-6989(88)80731-8","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1071-1072"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80731-8","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14341174","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Giacinto Bagetta, Elisabetta Priolo, Giuseppe Nistico
{"title":"Dopamine D-2 receptors in the ventral tegmental area mediate behavioural and electrocortical sleep of dopaminergic drugs in rats","authors":"Giacinto Bagetta, Elisabetta Priolo, Giuseppe Nistico","doi":"10.1016/S0031-6989(88)80741-0","DOIUrl":"10.1016/S0031-6989(88)80741-0","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1091-1092"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80741-0","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14042079","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
S. Amoroso , L. Annuziato , M. Taglialatela , G.F. Di Renzo , L.M.T. Canzoniero , G. Galizia , A. Marino
{"title":"Involvement of the Na+-H+ antiporter on the effect of protein kinase-C activation on dopamine synthesis in rat corpus striatum","authors":"S. Amoroso , L. Annuziato , M. Taglialatela , G.F. Di Renzo , L.M.T. Canzoniero , G. Galizia , A. Marino","doi":"10.1016/S0031-6989(88)80745-8","DOIUrl":"10.1016/S0031-6989(88)80745-8","url":null,"abstract":"","PeriodicalId":19810,"journal":{"name":"Pharmacological research communications","volume":"20 12","pages":"Pages 1099-1100"},"PeriodicalIF":0.0,"publicationDate":"1988-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/S0031-6989(88)80745-8","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"14042081","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}