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Chemistry of Heterocyclic Compounds最新文献

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Recent methods in the synthesis of chromeno[2,3-d]pyrimidines 合成色烯并[2,3-d]嘧啶的最新方法
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-04 DOI: 10.1007/s10593-024-03302-6
Ravi Varala, Mohan Kurra, Mohammed Amanullah, Mohamed Hussien, Mohammed Mujahid Alam
{"title":"Recent methods in the synthesis of chromeno[2,3-d]pyrimidines","authors":"Ravi Varala, Mohan Kurra, Mohammed Amanullah, Mohamed Hussien, Mohammed Mujahid Alam","doi":"10.1007/s10593-024-03302-6","DOIUrl":"https://doi.org/10.1007/s10593-024-03302-6","url":null,"abstract":"<p>The most recent synthetic methods to produce chromeno[2,3-<i>d</i>]pyrimidine derivatives from 2015 onwards are outlined, and this mini-review is divided into different chapters according to the type of the reaction.</p>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-04","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255661","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
A reaction of 2-carbonyl-substituted 1H-benzo[f]chromenes with N-arylamides of cyanoacetic acid 2-羰基取代的 1H-苯并[f]色烯与氰基乙酸的 N-芳基酰胺的反应
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-04 DOI: 10.1007/s10593-024-03312-4
Dmitry V. Osipov, Pavel E. Krasnikov, Alina A. Artemenko
{"title":"A reaction of 2-carbonyl-substituted 1H-benzo[f]chromenes with N-arylamides of cyanoacetic acid","authors":"Dmitry V. Osipov, Pavel E. Krasnikov, Alina A. Artemenko","doi":"10.1007/s10593-024-03312-4","DOIUrl":"https://doi.org/10.1007/s10593-024-03312-4","url":null,"abstract":"<p>A reaction of 2-trifluoroacetyl-1<i>H</i>-benzo[<i>f</i>]chromenes with <i>N</i>-arylamides of cyanoacetic acid led to the synthesis of a series of 2-oxo-6-trifluoromethylpyridine-3-carboxamides as products of a cascade of the carbo-Michael reaction, Thorpe–Ziegler cyclization, and Dimroth rearrangement. In the case of 1<i>H</i>-benzo[<i>f</i>]chromene-2-carbaldehydes, the corresponding Knoevenagel adducts were isolated.</p>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-04","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255441","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
The synthesis of ethyl 2-amino-1-(aryl)-5-(arylcarbamoyl)-6-oxo-1,6-dihydropyridine-3-carboxylates 2-氨基-1-(芳基)-5-(芳基氨基甲酰基)-6-氧代-1,6-二氢吡啶-3-羧酸乙酯的合成
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-04 DOI: 10.1007/s10593-024-03311-5
Anush Kh. Khachatryan, Katya A. Avagyan, Anush A. Sargsyan, Anait G. Simonyan, Henrik A. Panosyan, Armen G. Ayvazyan, Alik E. Badasyan
{"title":"The synthesis of ethyl 2-amino-1-(aryl)-5-(arylcarbamoyl)-6-oxo-1,6-dihydropyridine-3-carboxylates","authors":"Anush Kh. Khachatryan, Katya A. Avagyan, Anush A. Sargsyan, Anait G. Simonyan, Henrik A. Panosyan, Armen G. Ayvazyan, Alik E. Badasyan","doi":"10.1007/s10593-024-03311-5","DOIUrl":"https://doi.org/10.1007/s10593-024-03311-5","url":null,"abstract":"<p>A new method for the synthesis of previously unknown ethyl 2-amino-1-(aryl)-5-(arylcarbamoyl)-6-oxo-1,6-dihydropyridine-3-carboxylates by a reaction of ethyl 2-cyano-3-ethoxyacrylate with <i>N</i><sup>1</sup>,<i>N</i><sup>3</sup>-diarylmalonamides was developed. The antibacterial activity of some of the synthesized compounds was assayed.</p>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-04","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255655","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
The synthesis of furazano- and thiadiazolopyrazine steroids and their antiproliferative activity 呋喃并噻二唑并吡嗪类固醇的合成及其抗增殖活性
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-03 DOI: 10.1007/s10593-024-03319-x
Svetlana K. Vorontsova, Alexander M. Scherbakov, Mikhail E. Minyaev, Leonid G. Menchikov, Igor V. Zavarzin
{"title":"The synthesis of furazano- and thiadiazolopyrazine steroids and their antiproliferative activity","authors":"Svetlana K. Vorontsova, Alexander M. Scherbakov, Mikhail E. Minyaev, Leonid G. Menchikov, Igor V. Zavarzin","doi":"10.1007/s10593-024-03319-x","DOIUrl":"https://doi.org/10.1007/s10593-024-03319-x","url":null,"abstract":"<p>An effective method for the synthesis of heterocyclic steroids with the [1,2,5]oxadiazolo[3,4-<i>b</i>]pyrazine and [1,2,5]thiadiazolo[3,4-<i>b</i>]-pyrazine fragments was developed. The structure of the products was confirmed by X-ray structural analysis. The resulting compounds showed high antiproliferative activity against breast (MCF7) and prostate (22Rv1) cancer cells, which was not inferior to that of cisplatin and abiraterone acetate.</p>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-03","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255431","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
An efficient synthesis of (E)-3-[(dimethylamino)methylidene]furan-2(3H)-thiones and transamination reactions thereof (E)-3-[(二甲基氨基)亚甲基]呋喃-2(3H)-硫酮的高效合成及其转氨基反应
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-03 DOI: 10.1007/s10593-024-03309-z
Alexandra S. Tikhomolova, Zhanna V. Mamleeva, Alevtina Yu. Egorova
{"title":"An efficient synthesis of (E)-3-[(dimethylamino)methylidene]furan-2(3H)-thiones and transamination reactions thereof","authors":"Alexandra S. Tikhomolova, Zhanna V. Mamleeva, Alevtina Yu. Egorova","doi":"10.1007/s10593-024-03309-z","DOIUrl":"https://doi.org/10.1007/s10593-024-03309-z","url":null,"abstract":"<p>The conditions were developed and the optimal temperature regime was selected for a selective thionation of 5-aryl-3-[(dimethylamino)-methylidene]furan-2(3<i>H</i>)-ones with Lawesson's reagent. The stereochemistry of the synthesized 3-[(dimethylamino)methylidene]furan-2(3<i>H</i>)-thiones was established. Based on this, a number of 3-arylaminomethylidenefuran-2(3<i>H</i>)-thiones were synthesized <i>via</i> transamination reaction.</p>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-03","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255384","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis of 1,2-oxazine N-oxides via noncatalyzed hetero-Diels–Alder reactions of nitroalkenes (microreview) 通过硝基烯的非催化异狄尔斯-阿尔德反应合成 1,2-恶嗪 N-氧化物（微型综述）
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-06-03 DOI: 10.1007/s10593-024-03304-4
Radomir Jasiński
{"title":"Synthesis of 1,2-oxazine N-oxides via noncatalyzed hetero-Diels–Alder reactions of nitroalkenes (microreview)","authors":"Radomir Jasiński","doi":"10.1007/s10593-024-03304-4","DOIUrl":"https://doi.org/10.1007/s10593-024-03304-4","url":null,"abstract":"\u0000<figure></figure><p>In this microreview, the application of noncatalyzed hetero-Diels–Alder reaction (formally [4+2] cycloaddition) with participation of conjugated nitroalkenes and their analogs for easy and selective preparation of 1,2-oxazine <i>N</i>-oxides was reviewed on the basis of recent publications. It was found that the best described processes are realized with full regioselectivity as well as at mild temperatures. It is interesting, that in some cases of the title reactions, the stepwise mechanism of the formation of the six-membered heterocyclic ring is more possible than classic one-step mechanism.</p><figure><picture><source srcset=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03304-4/MediaObjects/10593_2024_3304_Figd_HTML.png?as=webp\" type=\"image/webp\"/><img alt=\"\" height=\"2\" loading=\"lazy\" src=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03304-4/MediaObjects/10593_2024_3304_Figd_HTML.png\" width=\"685\"/></picture></figure>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-06-03","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141255524","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis and reactivity of [1, 2, 5]thiadiazolo[3,4-b]pyridines and [1, 2, 5]selenadiazolo[3,4-b]pyridines (microreview) 1，2，5]噻二唑并[3，4-b]吡啶和[1，2，5]硒二唑并[3，4-b]吡啶的合成与反应性（微综述
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-04-12 DOI: 10.1007/s10593-024-03290-7
Maxim A. Bastrakov, Victoria V. Ivanova
{"title":"Synthesis and reactivity of [1, 2, 5]thiadiazolo[3,4-b]pyridines and [1, 2, 5]selenadiazolo[3,4-b]pyridines (microreview)","authors":"Maxim A. Bastrakov, Victoria V. Ivanova","doi":"10.1007/s10593-024-03290-7","DOIUrl":"https://doi.org/10.1007/s10593-024-03290-7","url":null,"abstract":"<p>\u0000<img alt=\"\" src=\"//media.springernature.com/lw234/springer-static/image/art%3A10.1007%2Fs10593-024-03290-7/MediaObjects/10593_2024_3290_Figc_HTML.png\" style=\"width:234px;max-width:none;\"/>\u0000The microreview covers the latest selected examples (2013–2024) on the synthesis and reactivity of [1, 2, 5]-thiadiazolo[3,4-<i>b</i>]pyridines and [1, 2, 5]selenadiazolo[3,4-<i>b</i>]pyridines. Their application is also discussed.</p><figure></figure>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-04-12","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"140566563","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis of fluorophores based on benzo[g]coumarin framework (microreview) 基于苯并[g]香豆素框架的荧光团合成（微综述）
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-04-11 DOI: 10.1007/s10593-024-03286-3
Ainur D. Sharapov, Ramil F. Fatykhov, Igor A. Khalymbadzha
{"title":"Synthesis of fluorophores based on benzo[g]coumarin framework (microreview)","authors":"Ainur D. Sharapov, Ramil F. Fatykhov, Igor A. Khalymbadzha","doi":"10.1007/s10593-024-03286-3","DOIUrl":"https://doi.org/10.1007/s10593-024-03286-3","url":null,"abstract":"\u0000<figure></figure><p>This microreview summarizes and analyzes literature for the years 2016–2023 on the construction of fluorophores based on benzo[<i>g</i>]coumarin backbone, which represent a push–pull system consisting of an annulated benzo and pyran rings. The main approaches to the synthesis of benzo[<i>g</i>]coumarins are condensation reactions, cyclization reactions, and pyran ring opening reactions followed by recyclization.</p><figure><picture><source srcset=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03286-3/MediaObjects/10593_2024_3286_Figd_HTML.png?as=webp\" type=\"image/webp\"/><img alt=\"\" height=\"2\" loading=\"lazy\" src=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03286-3/MediaObjects/10593_2024_3286_Figd_HTML.png\" width=\"685\"/></picture></figure>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-04-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"140566557","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis of carbonyl-containing nitrofurans (microreview) 含羰基的硝基呋喃的合成（微型综述）
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-04-11 DOI: 10.1007/s10593-024-03285-4
Kirill A. Gomonov, Vasilii V. Pelipko
{"title":"Synthesis of carbonyl-containing nitrofurans (microreview)","authors":"Kirill A. Gomonov, Vasilii V. Pelipko","doi":"10.1007/s10593-024-03285-4","DOIUrl":"https://doi.org/10.1007/s10593-024-03285-4","url":null,"abstract":"\u0000<figure></figure><p>This microreview analyzes and summarizes the most recent advances in the synthesis of carbonyl-containing nitrofurans, including methods of nitration, oxidation, and esterification of the corresponding furan derivatives, published since 2017.</p><figure><picture><source srcset=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03285-4/MediaObjects/10593_2024_3285_Figd_HTML.png?as=webp\" type=\"image/webp\"/><img alt=\"\" height=\"2\" loading=\"lazy\" src=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03285-4/MediaObjects/10593_2024_3285_Figd_HTML.png\" width=\"685\"/></picture></figure>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-04-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"140566911","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis of pyrrolizidine derivatives (microreview) 吡咯烷衍生物的合成（微型综述）
IF 1.5 4区 化学
Chemistry of Heterocyclic Compounds Pub Date : 2024-04-11 DOI: 10.1007/s10593-024-03287-2
Andrey V. Smolobochkin, Tanzilya S. Rizbayeva
{"title":"Synthesis of pyrrolizidine derivatives (microreview)","authors":"Andrey V. Smolobochkin, Tanzilya S. Rizbayeva","doi":"10.1007/s10593-024-03287-2","DOIUrl":"https://doi.org/10.1007/s10593-024-03287-2","url":null,"abstract":"\u0000<figure></figure><p>The review summarizes the methods of synthesis of pyrrolizidine (hexahydro-1<i>H</i>-pyrrolizine) derivatives published in the literature over the past five years. The methods can be conditionally divided into two major groups: synthesis from pyrrolidine derivatives and cyclization of acyclic precursors.</p><figure><picture><source srcset=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03287-2/MediaObjects/10593_2024_3287_Figd_HTML.png?as=webp\" type=\"image/webp\"/><img alt=\"\" height=\"2\" loading=\"lazy\" src=\"//media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs10593-024-03287-2/MediaObjects/10593_2024_3287_Figd_HTML.png\" width=\"685\"/></picture></figure>","PeriodicalId":9770,"journal":{"name":"Chemistry of Heterocyclic Compounds","volume":null,"pages":null},"PeriodicalIF":1.5,"publicationDate":"2024-04-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"140566470","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
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