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Synthesis and antifungal activities of bisbenzazole derivatives 双苯并唑衍生物的合成与抗真菌活性
Bioorganic and Medicinal Chemistry Reports Pub Date : 2024-08-09 DOI: 10.25135/acg.oc.2405.32434
Sule Gursoy, Dilara Ergun, Mehmet Abdullah Alagöz
{"title":"Synthesis and antifungal activities of bisbenzazole derivatives","authors":"Sule Gursoy, Dilara Ergun, Mehmet Abdullah Alagöz","doi":"10.25135/acg.oc.2405.32434","DOIUrl":"https://doi.org/10.25135/acg.oc.2405.32434","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2024-08-09","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"141922171","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Impact of COVID-19 on the thyroid gland in Iraqi females COVID-19 对伊拉克女性甲状腺的影响
Bioorganic and Medicinal Chemistry Reports Pub Date : 2024-02-14 DOI: 10.25135/bmcr.31.23.01.2775
R. Ersan, Kajeen H. Jasim, Noor Adnan Naeem, Lana Ziyad Sulayman, Rayan Sadiq, Nechervan Waheed, Jihan Hasan Jasim, Azheen Qasem
{"title":"Impact of COVID-19 on the thyroid gland in Iraqi females","authors":"R. Ersan, Kajeen H. Jasim, Noor Adnan Naeem, Lana Ziyad Sulayman, Rayan Sadiq, Nechervan Waheed, Jihan Hasan Jasim, Azheen Qasem","doi":"10.25135/bmcr.31.23.01.2775","DOIUrl":"https://doi.org/10.25135/bmcr.31.23.01.2775","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2024-02-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"139777550","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Impact of COVID-19 on the thyroid gland in Iraqi females COVID-19 对伊拉克女性甲状腺的影响
Bioorganic and Medicinal Chemistry Reports Pub Date : 2024-02-14 DOI: 10.25135/bmcr.31.23.01.2775
R. Ersan, Kajeen H. Jasim, Noor Adnan Naeem, Lana Ziyad Sulayman, Rayan Sadiq, Nechervan Waheed, Jihan Hasan Jasim, Azheen Qasem
{"title":"Impact of COVID-19 on the thyroid gland in Iraqi females","authors":"R. Ersan, Kajeen H. Jasim, Noor Adnan Naeem, Lana Ziyad Sulayman, Rayan Sadiq, Nechervan Waheed, Jihan Hasan Jasim, Azheen Qasem","doi":"10.25135/bmcr.31.23.01.2775","DOIUrl":"https://doi.org/10.25135/bmcr.31.23.01.2775","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2024-02-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"139837256","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Fluorinated benzimidazole derivatives: In vitro antimicrobial activity 氟化苯并咪唑衍生物:体外抗菌活性
Bioorganic and Medicinal Chemistry Reports Pub Date : 2023-07-31 DOI: 10.25135/bmcr.30.23.01.2692
Ronak Haj Ersan, Kajeen Jasim, Roaida Sadeeq, Soad Salim, Zina Fadhil, Somaya Mahmood
{"title":"Fluorinated benzimidazole derivatives: In vitro antimicrobial activity","authors":"Ronak Haj Ersan, Kajeen Jasim, Roaida Sadeeq, Soad Salim, Zina Fadhil, Somaya Mahmood","doi":"10.25135/bmcr.30.23.01.2692","DOIUrl":"https://doi.org/10.25135/bmcr.30.23.01.2692","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2023-07-31","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"135100236","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Fluorinated benzimidazole derivatives: In vitro antimicrobial activity 氟化苯并咪唑衍生物:体外抗菌活性
Bioorganic and Medicinal Chemistry Reports Pub Date : 2023-04-27 DOI: 10.25135/bmcr.30.23.01.2692x
R. Ersan, Kajeen H. Jasim, Roaida Sadeeq, Soad Salim, Zina Fadhil, Somaya Mahmood
{"title":"Fluorinated benzimidazole derivatives: In vitro antimicrobial activity","authors":"R. Ersan, Kajeen H. Jasim, Roaida Sadeeq, Soad Salim, Zina Fadhil, Somaya Mahmood","doi":"10.25135/bmcr.30.23.01.2692x","DOIUrl":"https://doi.org/10.25135/bmcr.30.23.01.2692x","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2023-04-27","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"88484768","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Comparing machine learning models for acetylcholine esterase inhibitors 比较乙酰胆碱酯酶抑制剂的机器学习模型
Bioorganic and Medicinal Chemistry Reports Pub Date : 2022-08-14 DOI: 10.25135/bmcr.29.22.06.2483
Mehmet Ali Yucel
{"title":"Comparing machine learning models for acetylcholine esterase inhibitors","authors":"Mehmet Ali Yucel","doi":"10.25135/bmcr.29.22.06.2483","DOIUrl":"https://doi.org/10.25135/bmcr.29.22.06.2483","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2022-08-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"86677119","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Cytotoxic activity evaluation of naphthalene substituted benzimidazole derivatives 萘取代苯并咪唑衍生物的细胞毒活性评价
Bioorganic and Medicinal Chemistry Reports Pub Date : 2022-05-17 DOI: 10.25135/acg.bmcr..28.2201.2322
R. Ersan, Kajeen H. Jasim, Haytham Sabeeh, K. Ahmed, Darya Abdulsatar, Shan Ali
{"title":"Cytotoxic activity evaluation of naphthalene substituted benzimidazole derivatives","authors":"R. Ersan, Kajeen H. Jasim, Haytham Sabeeh, K. Ahmed, Darya Abdulsatar, Shan Ali","doi":"10.25135/acg.bmcr..28.2201.2322","DOIUrl":"https://doi.org/10.25135/acg.bmcr..28.2201.2322","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2022-05-17","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"84098132","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Determination of Lidocaine HCl in commercially cream and injection forms by GC-FID method GC-FID法测定市售乳膏和注射剂中盐酸利多卡因的含量
Bioorganic and Medicinal Chemistry Reports Pub Date : 2022-05-15 DOI: 10.25135/bmcr.27.2204.2418
Y. Kadioglu, Alptug Atila
{"title":"Determination of Lidocaine HCl in commercially cream and injection forms by GC-FID method","authors":"Y. Kadioglu, Alptug Atila","doi":"10.25135/bmcr.27.2204.2418","DOIUrl":"https://doi.org/10.25135/bmcr.27.2204.2418","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2022-05-15","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"82314407","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Neuroprotective activity studies of some phenylacetamide derivatives bearing 1H-pyrazole or 1H-1,2,4-triazole 含1h -吡唑或1h -1,2,4-三唑的苯乙酰胺衍生物的神经保护活性研究
Bioorganic and Medicinal Chemistry Reports Pub Date : 2021-11-28 DOI: 10.25135/acg.bmcr.26.2111.2255
Merve Saylam, Ayse H. Tarikogullari, S. Yılmaz, P. Ballar Kirmizibayrak
{"title":"Neuroprotective activity studies of some phenylacetamide derivatives bearing 1H-pyrazole or 1H-1,2,4-triazole","authors":"Merve Saylam, Ayse H. Tarikogullari, S. Yılmaz, P. Ballar Kirmizibayrak","doi":"10.25135/acg.bmcr.26.2111.2255","DOIUrl":"https://doi.org/10.25135/acg.bmcr.26.2111.2255","url":null,"abstract":"","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2021-11-28","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"85542306","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis and biological evaluation of 1,3,5-triazine-substituted ureido benzenesulfonamides as antioxidant, acetylcholinesterase and butyrylcholinesterase inhibitors 1,3,5-三嗪取代脲基苯磺酰胺类抗氧化、乙酰胆碱酯酶和丁基胆碱酯酶抑制剂的合成及生物学评价
Bioorganic and Medicinal Chemistry Reports Pub Date : 2020-12-12 DOI: 10.25135/acg.bmcr.22.20.07.1706
Nebih Lolak, Muhammed Tuneğ, Asli E Dogan, M. Boğa, Suleyman Akocak
{"title":"Synthesis and biological evaluation of 1,3,5-triazine-substituted ureido benzenesulfonamides as antioxidant, acetylcholinesterase and butyrylcholinesterase inhibitors","authors":"Nebih Lolak, Muhammed Tuneğ, Asli E Dogan, M. Boğa, Suleyman Akocak","doi":"10.25135/acg.bmcr.22.20.07.1706","DOIUrl":"https://doi.org/10.25135/acg.bmcr.22.20.07.1706","url":null,"abstract":"A series of twenty 1,3,5-triazine-substituted ureido benzenesulfonamides 2 (a-e) and 3 (a-o) were re-synthesized and assayed for antioxidant properties by using several different methods including 1,1-diphenyl-2-picryl hydrazyl (DPPH) free radical scavenging assay, 2,2′-azino-bis-(3-ethylbenzothiazoline-6-sulfonic acid) (ABTS) cation radical decolarization assay, metal chelating and cupric reducing antioxidant capacity (CUPRAC) methods. The inhibitory effects of compounds on acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) enzymes have been also demonstrated. All compounds showed a greater antioxidant capacity against ABTS assay by having a more potent activity than the standards BHT, BHA and α-TOC. In general, all compounds were non susceptible to against AChE enzyme. On the other hand, several lead compounds were obtained from the current series against BChE enzyme. More specifically, compound 3m showed great inhibition profile against BChE with % inhibition value of 93.77, which is better than the standard drug galantamine (% inhibition value of 87.86).","PeriodicalId":8932,"journal":{"name":"Bioorganic and Medicinal Chemistry Reports","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2020-12-12","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"81472521","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 4
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