Francisca Cabrera-Escribano, Antonio Galera-Carrillo, R. Regalado, A. Franconetti, Óscar López-López
{"title":"Unprecedented Chitosan-derived Selenoureas","authors":"Francisca Cabrera-Escribano, Antonio Galera-Carrillo, R. Regalado, A. Franconetti, Óscar López-López","doi":"10.3390/ecsoc-22-05768","DOIUrl":"https://doi.org/10.3390/ecsoc-22-05768","url":null,"abstract":"","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"47 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123449354","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
M. Derita, Andrea B. J. Bracca, Iván Cortés, M. D. Liberto, T. Kaufman
{"title":"Cerium(III)-promoted synthesis of methoximes and preliminary results of their activity against phytopathogenic fungi","authors":"M. Derita, Andrea B. J. Bracca, Iván Cortés, M. D. Liberto, T. Kaufman","doi":"10.3390/ECSOC-22-05677","DOIUrl":"https://doi.org/10.3390/ECSOC-22-05677","url":null,"abstract":"The reaction between aromatic and aliphatic aldehydes and ketones with methoxylamine is promoted by cerium chloride. The antifungal activity of some methoxime derivatives against five postharvest phytopathogenic fungi, was examined, employing imazalil and carbendazim as positive controls, and the preliminary results are discussed. The target fungi were Rhizopus stolonifer , Botrytis cinerea, Penicillium digitatum, Penicillium italicum and Monilinia fructicola . These phytopathogens affect fruits worldwide, causing relevant economic damage. In all cases, minimum inhibitory concentrations and minimum fungicidal concentrations were obtained. Despite most of the simple compounds resulted inactive, preliminary results suggest that certain compounds display a structure-dependent activity which correlates with the length of the substituent attached to the oxime sp 2 carbon. _________________________________________________________________________","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"86 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"127099336","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
A. P. Nikalje, U. Nimbalkar, Julio A Seijas Vazquez, M. Vázquez-Tato
{"title":"Ultrasound-Assisted Facile Synthesis and Anticancer Evaluation of Novel N-(2-substituted phenyl-4-oxathiazolidine-3-carbonothioyl) benzamide","authors":"A. P. Nikalje, U. Nimbalkar, Julio A Seijas Vazquez, M. Vázquez-Tato","doi":"10.3390/ecsoc-22-05797","DOIUrl":"https://doi.org/10.3390/ecsoc-22-05797","url":null,"abstract":"","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"51 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"127422889","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Synthesis of an alkaline-earth metal organic frameworks (MOF) based on benzene-1,2,4,5 tetracarboxylic acid","authors":"F. Manteghi, Targol Rahimi Masale Nezhad","doi":"10.3390/ECSOC-22-05703","DOIUrl":"https://doi.org/10.3390/ECSOC-22-05703","url":null,"abstract":"","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"56 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"124548461","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Pyrrolidine analogs of arylceramide HPA-12","authors":"M. Zeman, Jozef Markus, D. Berkeš","doi":"10.3390/ECSOC-22-05673","DOIUrl":"https://doi.org/10.3390/ECSOC-22-05673","url":null,"abstract":": Conformational constraint is the usual way to modify the properties of bioactive molecules. In some cases, such modification improves their activity as well as their affinity for their biological target. At the beginning of the millennium, the ( R,R )-HPA-12 was found to be the first antagonist of ceramide transporter CERT, which has been identified as a key factor for the ER-to-Golgi trafficking of ceramides. Ten years later, we have revised the stereochemistry of the most active HPA-12 diastereomer to ( R , S )-diastereomer and developed synthesis of more potent alkyl substituted HPA-12 analogs. In this contribution, we would like to describe a straightforward approach to the enantiomerically pure constraint pyrrolidine analogs of both ( R,S )-HPA-12 and ( R,R )-HPA-12 starting from 3-substituted pyroglutamic acids easily accessible via our methodology. The results of the binding assays to the CERT protein will be discussed.","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"23 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"126061696","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
Fatima Lucio Martinez, J. M. Vila, Francisco Reigosa, P. Munín, J. M. Ortigueira, M. T. Pereira
{"title":"Synthesis and reactivity of a new type of crown ether thiosemicarbazone","authors":"Fatima Lucio Martinez, J. M. Vila, Francisco Reigosa, P. Munín, J. M. Ortigueira, M. T. Pereira","doi":"10.3390/ECSOC-22-05686","DOIUrl":"https://doi.org/10.3390/ECSOC-22-05686","url":null,"abstract":": Palladacycle compounds containing a crown-ether moiety in their structure have been scarcely studied in the past years, although they offer the possibility of combining the crown-ether application as sensors with the catalytic behavior of palladacycles. Maybe the reason for this is because they present a strong interaction with silica making the purification of the new products a difficult task. Nevertheless, in this communication we present the synthesis and characterization of a new palladacycle bearing a 15-crown-5-ether.","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"1 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"115927988","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Selective adsorption of a cationic dye by UiO-66-NH2","authors":"F. Manteghi, Fatemeh Varamini","doi":"10.3390/ECSOC-22-05695","DOIUrl":"https://doi.org/10.3390/ECSOC-22-05695","url":null,"abstract":"","PeriodicalId":448277,"journal":{"name":"Proceedings of The 22nd International Electronic Conference on Synthetic Organic Chemistry","volume":"34 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2018-11-14","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131496532","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}