A. Smirnov, E. Manakova, S. Gražulis, R. McKenna, D. Matulis
{"title":"Structures of Human Carbonic Anhydrases and Their Complexes with Inhibitors","authors":"A. Smirnov, E. Manakova, S. Gražulis, R. McKenna, D. Matulis","doi":"10.1007/978-3-030-12780-0_13","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_13","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"26 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"116762053","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Correlations Between Inhibitor Binding Thermodynamics and Co-crystal Structures with Carbonic Anhydrases","authors":"A. Smirnov, E. Manakova, D. Matulis","doi":"10.1007/978-3-030-12780-0_17","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_17","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"84 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"115332125","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"X-Ray Crystallographic Structures of High-Affinity and High-Selectivity Inhibitor Complexes with CA IX That Plays a Special Role in Cancer","authors":"K. Tārs, D. Matulis","doi":"10.1007/978-3-030-12780-0_14","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_14","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"13 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"125279476","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Organic Synthesis of Substituted Chlorinated Benzenesulfonamides as Selective Inhibitors of Several CA Isoforms","authors":"E. Čapkauskaitė, D. Matulis","doi":"10.1007/978-3-030-12780-0_10","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_10","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"1 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"130103724","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
V. Paketurytė, Asta Zubrienė, Wen-Yih Chen, S. Keller, M. Bastos, M. Todd, J. Ladbury, D. Matulis
{"title":"Inhibitor Binding to Carbonic Anhydrases by Isothermal Titration Calorimetry","authors":"V. Paketurytė, Asta Zubrienė, Wen-Yih Chen, S. Keller, M. Bastos, M. Todd, J. Ladbury, D. Matulis","doi":"10.1007/978-3-030-12780-0_6","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_6","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"46 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"128822628","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Inhibitor Binding to Carbonic Anhydrases by Fluorescent Thermal Shift Assay","authors":"V. Petrauskas, Asta Zubrienė, M. Todd, D. Matulis","doi":"10.1007/978-3-030-12780-0_5","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_5","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"56 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"117021508","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Clinical Trials Involving Carbonic Anhydrase IX as a Target for Cancer Diagnosis and Treatment","authors":"S. Grinceviciene, D. Matulis","doi":"10.1007/978-3-030-12780-0_22","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_22","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"36 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"116453499","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Organic Synthesis of Substituted Fluorinated Benzenesulfonamides as Selective Inhibitors of CA IX and Other Isoforms","authors":"V. Dudutienė, D. Matulis","doi":"10.1007/978-3-030-12780-0_11","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_11","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"15 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123940567","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Maps of Correlations Between Compound Chemical Structures and Thermodynamics of Binding to 12 Human Carbonic Anhydrases: Towards Isoform-Selective Inhibitors","authors":"Asta Zubrienė, Vaida Linkuvienė, D. Matulis","doi":"10.1007/978-3-030-12780-0_16","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_16","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"23 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"128698939","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Use of Carbonic Anhydrase IX Inhibitors for Selective Delivery of Attached Drugs to Solid Tumors","authors":"Spencer Gardeen, P. Low","doi":"10.1007/978-3-030-12780-0_19","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_19","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"1 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131224317","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}