Carbonic Anhydrase as Drug Target最新文献

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Structures of Human Carbonic Anhydrases and Their Complexes with Inhibitors 人碳酸酐酶的结构及其与抑制剂的配合物
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_13
A. Smirnov, E. Manakova, S. Gražulis, R. McKenna, D. Matulis
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引用次数: 1
Correlations Between Inhibitor Binding Thermodynamics and Co-crystal Structures with Carbonic Anhydrases 碳酸酐酶抑制剂结合热力学与共晶结构的关系
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_17
A. Smirnov, E. Manakova, D. Matulis
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引用次数: 1
X-Ray Crystallographic Structures of High-Affinity and High-Selectivity Inhibitor Complexes with CA IX That Plays a Special Role in Cancer 在癌症中起特殊作用的CA IX高亲和力和高选择性抑制剂配合物的x射线晶体结构
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_14
K. Tārs, D. Matulis
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引用次数: 1
Organic Synthesis of Substituted Chlorinated Benzenesulfonamides as Selective Inhibitors of Several CA Isoforms 取代氯代苯磺酰胺作为几种CA同工型选择性抑制剂的有机合成
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_10
E. Čapkauskaitė, D. Matulis
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引用次数: 1
Inhibitor Binding to Carbonic Anhydrases by Isothermal Titration Calorimetry 抑制剂与碳酸酐酶结合的等温滴定量热法
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_6
V. Paketurytė, Asta Zubrienė, Wen-Yih Chen, S. Keller, M. Bastos, M. Todd, J. Ladbury, D. Matulis
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引用次数: 3
Inhibitor Binding to Carbonic Anhydrases by Fluorescent Thermal Shift Assay 碳酸酐酶与抑制剂结合的荧光热移测定
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_5
V. Petrauskas, Asta Zubrienė, M. Todd, D. Matulis
{"title":"Inhibitor Binding to Carbonic Anhydrases by Fluorescent Thermal Shift Assay","authors":"V. Petrauskas, Asta Zubrienė, M. Todd, D. Matulis","doi":"10.1007/978-3-030-12780-0_5","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_5","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"56 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"117021508","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 11
Clinical Trials Involving Carbonic Anhydrase IX as a Target for Cancer Diagnosis and Treatment 碳酸酐酶IX作为癌症诊断和治疗靶点的临床试验
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_22
S. Grinceviciene, D. Matulis
{"title":"Clinical Trials Involving Carbonic Anhydrase IX as a Target for Cancer Diagnosis and Treatment","authors":"S. Grinceviciene, D. Matulis","doi":"10.1007/978-3-030-12780-0_22","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_22","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"36 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"116453499","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Organic Synthesis of Substituted Fluorinated Benzenesulfonamides as Selective Inhibitors of CA IX and Other Isoforms 取代氟化苯磺酰胺作为CA IX和其他同工异构体选择性抑制剂的有机合成
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_11
V. Dudutienė, D. Matulis
{"title":"Organic Synthesis of Substituted Fluorinated Benzenesulfonamides as Selective Inhibitors of CA IX and Other Isoforms","authors":"V. Dudutienė, D. Matulis","doi":"10.1007/978-3-030-12780-0_11","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_11","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"15 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"123940567","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Maps of Correlations Between Compound Chemical Structures and Thermodynamics of Binding to 12 Human Carbonic Anhydrases: Towards Isoform-Selective Inhibitors 化合物化学结构与12种人类碳酸酐酶结合热力学的相关性图:指向同型选择性抑制剂
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_16
Asta Zubrienė, Vaida Linkuvienė, D. Matulis
{"title":"Maps of Correlations Between Compound Chemical Structures and Thermodynamics of Binding to 12 Human Carbonic Anhydrases: Towards Isoform-Selective Inhibitors","authors":"Asta Zubrienė, Vaida Linkuvienė, D. Matulis","doi":"10.1007/978-3-030-12780-0_16","DOIUrl":"https://doi.org/10.1007/978-3-030-12780-0_16","url":null,"abstract":"","PeriodicalId":444527,"journal":{"name":"Carbonic Anhydrase as Drug Target","volume":"23 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"1900-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"128698939","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Use of Carbonic Anhydrase IX Inhibitors for Selective Delivery of Attached Drugs to Solid Tumors 使用碳酸酐酶IX抑制剂选择性递送附着药物到实体肿瘤
Carbonic Anhydrase as Drug Target Pub Date : 1900-01-01 DOI: 10.1007/978-3-030-12780-0_19
Spencer Gardeen, P. Low
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引用次数: 1
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