Progress in medicinal chemistry最新文献

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Glucokinase. Preface. 葡糖激酶。前言。
Progress in medicinal chemistry Pub Date : 2013-01-01 DOI: 10.1016/B978-0-444-62652-3.10000-6
Geoff Lawton, David R Witty
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引用次数: 0
Antimalarial drug discovery: recent progress and future directions. 抗疟药物的发现:最新进展和未来方向。
Progress in medicinal chemistry Pub Date : 2013-01-01 DOI: 10.1016/B978-0-444-62652-3.00003-X
Félix Calderón, David M Wilson, Francisco-Javier Gamo
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引用次数: 31
Medicinal chemistry of glucagon-like peptide receptor agonists. 胰高血糖素样肽受体激动剂的药物化学。
Progress in medicinal chemistry Pub Date : 2013-01-01 DOI: 10.1016/B978-0-444-62652-3.00002-8
Lyn H Jones, David A Price
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引用次数: 12
Property-based design in the optimisation of benzamide glucokinase activators: from hit to clinic. 苯甲酰胺葡萄糖激酶活化剂优化中的基于性能的设计:从hit到临床。
Progress in medicinal chemistry Pub Date : 2013-01-01 DOI: 10.1016/B978-0-444-62652-3.00001-6
Darren McKerrecher, Michael J Waring
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引用次数: 4
Hematopoietic prostaglandin D synthase inhibitors. 造血前列腺素D合成酶抑制剂。
Progress in medicinal chemistry Pub Date : 2012-01-01 DOI: 10.1016/B978-0-12-396493-9.00004-2
Sukanthini Thurairatnam
{"title":"Hematopoietic prostaglandin D synthase inhibitors.","authors":"Sukanthini Thurairatnam","doi":"10.1016/B978-0-12-396493-9.00004-2","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00004-2","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"97-133"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00004-2","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171225","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 20
TRPV1 antagonists: clinical setbacks and prospects for future development. TRPV1拮抗剂:临床挫折及未来发展前景
Progress in medicinal chemistry Pub Date : 2012-01-01 DOI: 10.1016/B978-0-12-396493-9.00002-9
Michael E Kort, Philip R Kym
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引用次数: 57
Multivalent dual pharmacology muscarinic antagonist and β₂ agonist (MABA) molecules for the treatment of COPD. 多价双重药理毒蕈碱拮抗剂和β 2激动剂(MABA)分子治疗COPD。
Progress in medicinal chemistry Pub Date : 2012-01-01 DOI: 10.1016/B978-0-12-396493-9.00003-0
Adam D Hughes, Alexander McNamara, Tod Steinfeld
{"title":"Multivalent dual pharmacology muscarinic antagonist and β₂ agonist (MABA) molecules for the treatment of COPD.","authors":"Adam D Hughes, Alexander McNamara, Tod Steinfeld","doi":"10.1016/B978-0-12-396493-9.00003-0","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00003-0","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"71-95"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00003-0","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171224","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 25
Small molecule bromodomain inhibitors: extending the druggable genome. 小分子溴结构域抑制剂:扩展可药物基因组。
Progress in medicinal chemistry Pub Date : 2012-01-01 DOI: 10.1016/B978-0-12-396493-9.00001-7
Chun-Wa Chung
{"title":"Small molecule bromodomain inhibitors: extending the druggable genome.","authors":"Chun-Wa Chung","doi":"10.1016/B978-0-12-396493-9.00001-7","DOIUrl":"https://doi.org/10.1016/B978-0-12-396493-9.00001-7","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"51 ","pages":"1-55"},"PeriodicalIF":0.0,"publicationDate":"2012-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-396493-9.00001-7","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"40171222","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 43
The large scale restructuring of pharmaceutical company research function. Preface. 医药企业研究职能的大规模重组。前言。
Progress in medicinal chemistry Pub Date : 2012-01-01 DOI: 10.1016/B978-0-12-396493-9.00005-4
G Lawton, David R Witty
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引用次数: 0
Designing drugs to avoid toxicity. 设计药物以避免毒性。
Progress in medicinal chemistry Pub Date : 2011-01-01 DOI: 10.1016/B978-0-12-381290-2.00001-X
Graham F Smith
{"title":"Designing drugs to avoid toxicity.","authors":"Graham F Smith","doi":"10.1016/B978-0-12-381290-2.00001-X","DOIUrl":"https://doi.org/10.1016/B978-0-12-381290-2.00001-X","url":null,"abstract":"","PeriodicalId":20755,"journal":{"name":"Progress in medicinal chemistry","volume":"50 ","pages":"1-47"},"PeriodicalIF":0.0,"publicationDate":"2011-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://sci-hub-pdf.com/10.1016/B978-0-12-381290-2.00001-X","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"29667943","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 85
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