ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology最新文献

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Structure based approaches on fentanyl template to design novel mu opioid modulators 基于芬太尼模板的结构方法设计新型mu阿片调节剂
Rohini S. Ople, Haoqing Wang, Qiongyu Li, Ben Polacco, Sarah M. Bernhard, K. Appourchaux, Sashrik Sribhashyam, S. Eans, Ruth Huttenhain, Jay P. McLaughlin, B. Kobilka, S. Majumdar
{"title":"Structure based approaches on fentanyl template to design novel mu opioid modulators","authors":"Rohini S. Ople, Haoqing Wang, Qiongyu Li, Ben Polacco, Sarah M. Bernhard, K. Appourchaux, Sashrik Sribhashyam, S. Eans, Ruth Huttenhain, Jay P. McLaughlin, B. Kobilka, S. Majumdar","doi":"10.1124/jpet.122.527690","DOIUrl":"https://doi.org/10.1124/jpet.122.527690","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"26 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"115371372","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Calmodulin Dependent Protein Kinase II: An Effector in the Signaling Pathway of Antidepressant-like Behavior Elicited by Ketamine in Combination with Melatonin 钙调素依赖性蛋白激酶II:氯胺酮与褪黑激素联合引发的抗抑郁样行为信号通路中的效应物
G. Benítez-King, Armida Miranda-Riestra, R. Estrada-Reyes, C. Trueta, Jesús Argueta, Julián Oikawa-Sala, L. A. Constantino-Jonapa, Montserrat G Cercós
{"title":"Calmodulin Dependent Protein Kinase II: An Effector in the Signaling Pathway of Antidepressant-like Behavior Elicited by Ketamine in Combination with Melatonin","authors":"G. Benítez-King, Armida Miranda-Riestra, R. Estrada-Reyes, C. Trueta, Jesús Argueta, Julián Oikawa-Sala, L. A. Constantino-Jonapa, Montserrat G Cercós","doi":"10.1124/jpet.122.215840","DOIUrl":"https://doi.org/10.1124/jpet.122.215840","url":null,"abstract":"ID","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"67 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"117243706","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Mediation Analysis Reveals that Opioid-Induced Sleep Disruption is Partially Mediated by Increased Motor Activity in C57BL/6J (B6) Mice 中介分析显示阿片类药物引起的睡眠中断部分是由C57BL/6J (B6)小鼠运动活动增加介导的
Diana Zebadúa Unzaga, Xiaojuan Zhu, J. Price, Michael A. Oneil, R. Lydic, H. Baghdoyan
{"title":"Mediation Analysis Reveals that Opioid-Induced Sleep Disruption is Partially Mediated by Increased Motor Activity in C57BL/6J (B6) Mice","authors":"Diana Zebadúa Unzaga, Xiaojuan Zhu, J. Price, Michael A. Oneil, R. Lydic, H. Baghdoyan","doi":"10.1124/jpet.122.192550","DOIUrl":"https://doi.org/10.1124/jpet.122.192550","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"115 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"120936087","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Comparison of the mu-opioid receptor antagonists methocinnamox (MCAM) and naloxone to reverse the ventilatory-depressant effects of fentanyl and heroin in male rats 莫阿片受体拮抗剂甲氧西那莫(MCAM)和纳洛酮逆转芬太尼和海洛因对雄性大鼠通气抑制作用的比较
T. Hiranita, Nicholas P. Ho, C. France
{"title":"Comparison of the mu-opioid receptor antagonists methocinnamox (MCAM) and naloxone to reverse the ventilatory-depressant effects of fentanyl and heroin in male rats","authors":"T. Hiranita, Nicholas P. Ho, C. France","doi":"10.1124/jpet.122.155410","DOIUrl":"https://doi.org/10.1124/jpet.122.155410","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"157 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"121017537","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Gain Modulation by Mouse Prefrontal Cortex Diminishes Fentanyl-Induced Respiratory Depression 小鼠前额叶皮层的增益调节减轻芬太尼诱导的呼吸抑制
Daniel P. Woods, Ryan S. Herzog, Qi Sun, Zachary T. Glovak, H. Baghdoyan, R. Lydic
{"title":"Gain Modulation by Mouse Prefrontal Cortex Diminishes Fentanyl-Induced Respiratory Depression","authors":"Daniel P. Woods, Ryan S. Herzog, Qi Sun, Zachary T. Glovak, H. Baghdoyan, R. Lydic","doi":"10.1124/jpet.122.530000","DOIUrl":"https://doi.org/10.1124/jpet.122.530000","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"78 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"126292305","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Effectiveness of GPR171 Agonist with Morphine and Identification of GPR171 Signaling Profile 吗啡联合GPR171激动剂的有效性及GPR171信号谱的鉴定
Callie Porter, E. Bobeck
{"title":"Effectiveness of GPR171 Agonist with Morphine and Identification of GPR171 Signaling Profile","authors":"Callie Porter, E. Bobeck","doi":"10.1124/jpet.122.217300","DOIUrl":"https://doi.org/10.1124/jpet.122.217300","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"50 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"125487979","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Prenatal Stress Alters Transcription of NMDA Receptors in the Frontal Cortex and Hippocampus 产前应激改变额叶皮质和海马中NMDA受体的转录
Tristram Buck, M. Sodhi
{"title":"Prenatal Stress Alters Transcription of NMDA Receptors in the Frontal Cortex and Hippocampus","authors":"Tristram Buck, M. Sodhi","doi":"10.1124/jpet.122.258850","DOIUrl":"https://doi.org/10.1124/jpet.122.258850","url":null,"abstract":"Abstract","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"118 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"134139716","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Coronaridine Congeners Attenuate Fentanyl Seeking During Prolonged Abstinence, Possibly Through Inhibiting Dopamine Release in the Nucleus Accumbens 冠状萘啶同系物可能通过抑制伏隔核多巴胺释放,在长期戒断期间减弱芬太尼寻求
Jacob D. Layne, Mason J. Hochstetler, Brandon M. Curry, Benjamin M. Williams, Christina A. Small, S. Steffensen, H. Arias, Craig T. Werner
{"title":"Coronaridine Congeners Attenuate Fentanyl Seeking During Prolonged Abstinence, Possibly Through Inhibiting Dopamine Release in the Nucleus Accumbens","authors":"Jacob D. Layne, Mason J. Hochstetler, Brandon M. Curry, Benjamin M. Williams, Christina A. Small, S. Steffensen, H. Arias, Craig T. Werner","doi":"10.1124/jpet.122.542600","DOIUrl":"https://doi.org/10.1124/jpet.122.542600","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"6 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"131853674","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Presynaptic Regulation of Monoamine Release in the Dorsal Raphe Nucleus by Alpha2-adrenergic Receptors α 2-肾上腺素能受体对中缝背核单胺释放的突触前调节
Aleigha Gugel, Stephanie C. Gantz
{"title":"Presynaptic Regulation of Monoamine Release in the Dorsal Raphe Nucleus by Alpha2-adrenergic Receptors","authors":"Aleigha Gugel, Stephanie C. Gantz","doi":"10.1124/jpet.122.232630","DOIUrl":"https://doi.org/10.1124/jpet.122.232630","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"33 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"115927118","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Interactions between Biological Sex and Hormonal Cycles in Stimulant Effects on Motor Behavior 生理性别和激素周期对运动行为刺激作用的相互作用
Abigail Carr, J. Tat, E. Calipari, Kristy R. Erickson
{"title":"Interactions between Biological Sex and Hormonal Cycles in Stimulant Effects on Motor Behavior","authors":"Abigail Carr, J. Tat, E. Calipari, Kristy R. Erickson","doi":"10.1124/jpet.122.189820","DOIUrl":"https://doi.org/10.1124/jpet.122.189820","url":null,"abstract":"","PeriodicalId":177194,"journal":{"name":"ASPET 2023 Annual Meeting Abstract - Central Nervous System Pharmacology - Neuropharmacology","volume":"9 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-05-18","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"124418834","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":0,"RegionCategory":"","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
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