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Advances on Catalytic Approaches towards the Synthesis of Quinoline Derivatives Using Povarov Reaction 用Povarov反应催化合成喹啉衍生物的研究进展
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/rev-23-1004
Chandi C. Malakar, K. Kant, Sourav Banerjee, Chandresh K. Patel, S. Kalita, N. Aljaar, Reetu Reetu, Priyadarshini Naik
{"title":"Advances on Catalytic Approaches towards the Synthesis of Quinoline Derivatives Using Povarov Reaction","authors":"Chandi C. Malakar, K. Kant, Sourav Banerjee, Chandresh K. Patel, S. Kalita, N. Aljaar, Reetu Reetu, Priyadarshini Naik","doi":"10.3987/rev-23-1004","DOIUrl":"https://doi.org/10.3987/rev-23-1004","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70752286","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Chiral Benzimidazolium N-Heterocyclic Carbene Ligands with Hydroxyamide- or Hydroxyalkyl-Functionalized Wingtip for Cu-Catalyzed Asymmetric Allylic Alkylation 手性苯并咪唑n杂环卡宾配体与羟基酰胺或羟基烷基功能化翼尖铜催化的不对称烯丙基烷基化
4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14880
Satoshi Sakaguchi, Shota Takayanagi
{"title":"Chiral Benzimidazolium N-Heterocyclic Carbene Ligands with Hydroxyamide- or Hydroxyalkyl-Functionalized Wingtip for Cu-Catalyzed Asymmetric Allylic Alkylation","authors":"Satoshi Sakaguchi, Shota Takayanagi","doi":"10.3987/com-23-14880","DOIUrl":"https://doi.org/10.3987/com-23-14880","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"135441411","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Efficient Synthesis of Quinazoline-2,4(1H,3H)-Diones from 2-Aminobenzonitriles and Co2 Catalyzed by 2-Hydroxypyridine Anion-Based Ionic Liquid at Atmospheric Pressure 常压下2-羟基吡啶阴离子液体催化2-氨基苯并腈和Co2高效合成喹唑啉-2,4(1H,3H)-二酮
4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14892
Qi Feng, Lele Li, Jiayi Jin, Wanyao Hu, Jiayi Huang
{"title":"Efficient Synthesis of Quinazoline-2,4(1H,3H)-Diones from 2-Aminobenzonitriles and Co2 Catalyzed by 2-Hydroxypyridine Anion-Based Ionic Liquid at Atmospheric Pressure","authors":"Qi Feng, Lele Li, Jiayi Jin, Wanyao Hu, Jiayi Huang","doi":"10.3987/com-23-14892","DOIUrl":"https://doi.org/10.3987/com-23-14892","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.0,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"136004454","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis and Antitumor Activity of Heterocylic Aurone and Its Analogue Indanone Derivatives 杂环金酮及其类似物吲哚酮衍生物的合成及抗肿瘤活性研究
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-22-14764
H. Akber Aisa, C. Niu, Heng Wu, Ayitila Maimaitijiang, Dan-Jie Tang, Baoxing Xie
{"title":"Synthesis and Antitumor Activity of Heterocylic Aurone and Its Analogue Indanone Derivatives","authors":"H. Akber Aisa, C. Niu, Heng Wu, Ayitila Maimaitijiang, Dan-Jie Tang, Baoxing Xie","doi":"10.3987/com-22-14764","DOIUrl":"https://doi.org/10.3987/com-22-14764","url":null,"abstract":"– Based on non-classical bioisosterism and the rule of alkene insertion, thirty-five heterocyclic aurones and its analogue indanones derivatives were designed and synthesized. They were evaluated for inhibitory activity against HELA, HT-29 and A549 and HepG2 human cancer cell lines. Among them, twenty-five compounds exhibited moderate to excellent antitumor activity. The minimum value of IC 50 was 1.649±0.083 μM (compound B1 ). The SAR showed that aurone with B ring as aromatic heterocycles such as 4-bromothiophene, quinoline, carbazole and indanone derivatives and some or indanone were more potent than others. Besides, the introduction of acetylated glycosides was beneficial to the activity. Compounds A1 , B1 , C5 , C8 , C10 , C11 , C12 and D1 were promising antitumor agents. Among them, compounds molecular docking studies were performed between B1 , C8 and potential targets Aurora B (PBD: 2BFY). On the basis, the chemical and physical properties, as well as ADMET of active compounds were predicted and analyzed. And it showed that most of compounds had good pharmacokinetic profiles and high safety profiles","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70398643","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 1
Supramolecular Self-Assembly Based on Symmetric Tetramethyl-Substituted Cucurbit[6]uril and Small Aromatic Amines 基于对称四甲基取代葫芦b[6]和小芳胺的超分子自组装
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-22-14771
Qianjun Zhang, Lin Zhang, Jun Zheng, Xuan Wang, Z. Tao
{"title":"Supramolecular Self-Assembly Based on Symmetric Tetramethyl-Substituted Cucurbit[6]uril and Small Aromatic Amines","authors":"Qianjun Zhang, Lin Zhang, Jun Zheng, Xuan Wang, Z. Tao","doi":"10.3987/com-22-14771","DOIUrl":"https://doi.org/10.3987/com-22-14771","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70398819","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
12-epi-Briacavatolide B, a New Briarane Diterpenoid from the Octocoral Briareum stechei 12-epi-Briacavatolide B，一种新的briacavatolide二萜类化合物
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-22-14792
P. Sung, Chia-Jung Liu, Hsin-Tzu Liu, Thanh Hao Huynh, Z. Wen, Chia-Ching Liaw, Jih-Jung Chen, J. Su
{"title":"12-epi-Briacavatolide B, a New Briarane Diterpenoid from the Octocoral Briareum stechei","authors":"P. Sung, Chia-Jung Liu, Hsin-Tzu Liu, Thanh Hao Huynh, Z. Wen, Chia-Ching Liaw, Jih-Jung Chen, J. Su","doi":"10.3987/com-22-14792","DOIUrl":"https://doi.org/10.3987/com-22-14792","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70399051","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Sulfate Radical Anion (SO4˙ˉ) Mediated Degradation of Some Over-the-Counter Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) at Neutral Ph in Aqueous Environment 硫酸根阴离子(SO4˙离子)介导的非处方非甾体抗炎药(NSAIDs)在水环境中性Ph下的降解
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14804
Joydev K. Laha, Neelam Manral, Sagar Badoni, Mandeep Kaur Hunjan, Upma Gulati
{"title":"Sulfate Radical Anion (SO4˙ˉ) Mediated Degradation of Some Over-the-Counter Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) at Neutral Ph in Aqueous Environment","authors":"Joydev K. Laha, Neelam Manral, Sagar Badoni, Mandeep Kaur Hunjan, Upma Gulati","doi":"10.3987/com-23-14804","DOIUrl":"https://doi.org/10.3987/com-23-14804","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70400340","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
One-Pot Synthesis of Carbazoles by a Domino Reaction Using Microwave Heating and Antiproliferative Activities of Constituents from Murraya Plants Against Cancer Stem Cells 微波加热多米诺反应一锅法合成咔唑及其对肿瘤干细胞的抗增殖活性
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14816
Seikou Nakamura, Kouta Ugawa, Momona Nakao, Chikako Sawada, Takahiro Matsumoto, Takahiro Kitagawa, Yutaro Ohki, Kousuke Araki
{"title":"One-Pot Synthesis of Carbazoles by a Domino Reaction Using Microwave Heating and Antiproliferative Activities of Constituents from Murraya Plants Against Cancer Stem Cells","authors":"Seikou Nakamura, Kouta Ugawa, Momona Nakao, Chikako Sawada, Takahiro Matsumoto, Takahiro Kitagawa, Yutaro Ohki, Kousuke Araki","doi":"10.3987/com-23-14816","DOIUrl":"https://doi.org/10.3987/com-23-14816","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70400586","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Synthesis of 2-Anilino-2,4,4,6,6-pentachlorocyclotriphosphazenes (N3P3Cl5(NAr(R))) 2-苯胺-2,4,4,6,6-五氯环三磷杂烯(N3P3Cl5(NAr(R)))的合成
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14849
M. Kuroboshi*, Ryota Takahashi, Hideo Tanaka
{"title":"Synthesis of 2-Anilino-2,4,4,6,6-pentachlorocyclotriphosphazenes (N3P3Cl5(NAr(R)))","authors":"M. Kuroboshi*, Ryota Takahashi, Hideo Tanaka","doi":"10.3987/com-23-14849","DOIUrl":"https://doi.org/10.3987/com-23-14849","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70401319","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
Fischer Glycosidation Using Organotitanium Catalyst Orgatix 有机钛催化剂的Fischer糖苷化
IF 0.6 4区 化学
Heterocycles Pub Date : 2023-01-01 DOI: 10.3987/com-23-14866
Minoru Izumi, Nana Yanagida, Keita Kato, Mako Matsushita
{"title":"Fischer Glycosidation Using Organotitanium Catalyst Orgatix","authors":"Minoru Izumi, Nana Yanagida, Keita Kato, Mako Matsushita","doi":"10.3987/com-23-14866","DOIUrl":"https://doi.org/10.3987/com-23-14866","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":null,"pages":null},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70401474","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
引用次数: 0
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