HeterocyclesPub Date : 2023-01-01DOI: 10.3987/com-23-14824
Longjia Yan, Yaqing Zuo, Kehui Chen, Ying Xu, Y. Le
{"title":"Synthesis and Biological Evaluation of 5-Methylpyrimidine Derivatives as Dual Inhibitors of EGFR and Src for Cancer Treatment","authors":"Longjia Yan, Yaqing Zuo, Kehui Chen, Ying Xu, Y. Le","doi":"10.3987/com-23-14824","DOIUrl":"https://doi.org/10.3987/com-23-14824","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"1 1","pages":""},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70401116","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
HeterocyclesPub Date : 2023-01-01DOI: 10.3987/com-23-14837
H. Reissig, Morshed Alam Chowdhury
{"title":"Asymmetric Synthesis of the Unnatural Enantiomer of Codonopsinine and a Stereoisomer via Alkoxyallenes","authors":"H. Reissig, Morshed Alam Chowdhury","doi":"10.3987/com-23-14837","DOIUrl":"https://doi.org/10.3987/com-23-14837","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"1 1","pages":""},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70401224","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
HeterocyclesPub Date : 2023-01-01DOI: 10.3987/com-23-14872
N. Lu, Chengxia Miao, Xiaozheng Lan
{"title":"Theoretical Investigation of Cp*CO(III)-Mediated Regioselective [4 + 2]-Annulation of N-Chlorobenzamide with Vinyl Acetate for the Synthesis of Isoquinolone","authors":"N. Lu, Chengxia Miao, Xiaozheng Lan","doi":"10.3987/com-23-14872","DOIUrl":"https://doi.org/10.3987/com-23-14872","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"1 1","pages":""},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70401878","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
HeterocyclesPub Date : 2023-01-01DOI: 10.3987/rev-22-1001
H. Muraoka, S. Ogawa
{"title":"1,3,5-Triazine-Cored Star-Shaped (D-π)3-A Molecules Based on 2,4,6-Tris(5-Arylthiophen-2-Yl)-1,3,5-Triazine","authors":"H. Muraoka, S. Ogawa","doi":"10.3987/rev-22-1001","DOIUrl":"https://doi.org/10.3987/rev-22-1001","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"1 1","pages":""},"PeriodicalIF":0.6,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"70751360","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
{"title":"Facile Preparation of the Nootropic Agent IDRA-21 and Related Heterocycles via a One-Pot Iron-Mediated Redox Annulation","authors":"Kyosuke Kaneda, Hirotoshi Kabasawa, Syun Nabeki, Uki Matsui, Hiroki Sugiyama, Takehiro Yamagishi","doi":"10.3987/com-23-14893","DOIUrl":"https://doi.org/10.3987/com-23-14893","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"142 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"135440089","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
HeterocyclesPub Date : 2023-01-01DOI: 10.3987/rev-23-1014
Hala Bakr El-Nassan, Mohamed Osama Mousa, Mina Emad Adly, Amr Mohamed Mahmoud
{"title":"A Review on the Biological Activity of β-Carboline Derivatives","authors":"Hala Bakr El-Nassan, Mohamed Osama Mousa, Mina Emad Adly, Amr Mohamed Mahmoud","doi":"10.3987/rev-23-1014","DOIUrl":"https://doi.org/10.3987/rev-23-1014","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"33 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"135508711","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}
HeterocyclesPub Date : 2023-01-01DOI: 10.3987/rev-23-1013
Masahiro Nagase, Masatoshi Murakata
{"title":"Strategy for the Synthesis of C-Aryl Glucosides as Sodium Glucose Cotransporter 2 Inhibitors","authors":"Masahiro Nagase, Masatoshi Murakata","doi":"10.3987/rev-23-1013","DOIUrl":"https://doi.org/10.3987/rev-23-1013","url":null,"abstract":"","PeriodicalId":13166,"journal":{"name":"Heterocycles","volume":"26 1","pages":"0"},"PeriodicalIF":0.0,"publicationDate":"2023-01-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":null,"resultStr":null,"platform":"Semanticscholar","paperid":"135508712","PeriodicalName":null,"FirstCategoryId":null,"ListUrlMain":null,"RegionNum":4,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":"","EPubDate":null,"PubModel":null,"JCR":null,"JCRName":null,"Score":null,"Total":0}