由磺酰叠氮化物和炔烃合成具有生物活性的1-磺酰基-1,2,3-三唑：综述

IF 2.1 3区化学 Q3 CHEMISTRY, MULTIDISCIPLINARY

Journal of Sulfur Chemistry Pub Date : 2023-06-01 DOI:10.1080/17415993.2022.2149266

Mustafa M. Kadhim , Evan Abdulkareem Mahmood , Mohammad Reza Poor Heravi , Somayeh Soleimani-Amiri , Abdol Ghaffar Ebadi , Esmail Vessally

{"title":"由磺酰叠氮化物和炔烃合成具有生物活性的1-磺酰基-1,2,3-三唑：综述","authors":"Mustafa M. Kadhim , Evan Abdulkareem Mahmood , Mohammad Reza Poor Heravi , Somayeh Soleimani-Amiri , Abdol Ghaffar Ebadi , Esmail Vessally","doi":"10.1080/17415993.2022.2149266","DOIUrl":null,"url":null,"abstract":"<div><p>In this review, we spotlight the methods for the direct synthesis of synthetically and biologically important 1-sulfonyl-1, 2, 3-triazoles <em>via</em> [3+2] cycloaddition between easily available terminal alkynes and sulfonyl azides. The review is divided into two major sections. The first section focuses exclusively on the synthesis of 1-(<em>N</em>-sulfonyl)-4-substituted 1,2,3-triazoles, while the second section will discuss preparation of 1-(<em>N</em>-sulfonyl)-5-substituted 1,2,3-triazole derivatives.</p></div>","PeriodicalId":17081,"journal":{"name":"Journal of Sulfur Chemistry","volume":"44 3","pages":"Pages 377-391"},"PeriodicalIF":2.1000,"publicationDate":"2023-06-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":"1","resultStr":"{\"title\":\"The synthesis of biologically active 1-sulfonyl-1, 2, 3-triazoles from sulfonyl azides and alkynes: a focus review\",\"authors\":\"Mustafa M. Kadhim , Evan Abdulkareem Mahmood , Mohammad Reza Poor Heravi , Somayeh Soleimani-Amiri , Abdol Ghaffar Ebadi , Esmail Vessally\",\"doi\":\"10.1080/17415993.2022.2149266\",\"DOIUrl\":null,\"url\":null,\"abstract\":\"<div><p>In this review, we spotlight the methods for the direct synthesis of synthetically and biologically important 1-sulfonyl-1, 2, 3-triazoles <em>via</em> [3+2] cycloaddition between easily available terminal alkynes and sulfonyl azides. The review is divided into two major sections. The first section focuses exclusively on the synthesis of 1-(<em>N</em>-sulfonyl)-4-substituted 1,2,3-triazoles, while the second section will discuss preparation of 1-(<em>N</em>-sulfonyl)-5-substituted 1,2,3-triazole derivatives.</p></div>\",\"PeriodicalId\":17081,\"journal\":{\"name\":\"Journal of Sulfur Chemistry\",\"volume\":\"44 3\",\"pages\":\"Pages 377-391\"},\"PeriodicalIF\":2.1000,\"publicationDate\":\"2023-06-01\",\"publicationTypes\":\"Journal Article\",\"fieldsOfStudy\":null,\"isOpenAccess\":false,\"openAccessPdf\":\"\",\"citationCount\":\"1\",\"resultStr\":null,\"platform\":\"Semanticscholar\",\"paperid\":null,\"PeriodicalName\":\"Journal of Sulfur Chemistry\",\"FirstCategoryId\":\"92\",\"ListUrlMain\":\"https://www.sciencedirect.com/org/science/article/pii/S1741599323000053\",\"RegionNum\":3,\"RegionCategory\":\"化学\",\"ArticlePicture\":[],\"TitleCN\":null,\"AbstractTextCN\":null,\"PMCID\":null,\"EPubDate\":\"\",\"PubModel\":\"\",\"JCR\":\"Q3\",\"JCRName\":\"CHEMISTRY, MULTIDISCIPLINARY\",\"Score\":null,\"Total\":0}","platform":"Semanticscholar","paperid":null,"PeriodicalName":"Journal of Sulfur Chemistry","FirstCategoryId":"92","ListUrlMain":"https://www.sciencedirect.com/org/science/article/pii/S1741599323000053","RegionNum":3,"RegionCategory":"化学","ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":null,"EPubDate":"","PubModel":"","JCR":"Q3","JCRName":"CHEMISTRY, MULTIDISCIPLINARY","Score":null,"Total":0}

引用次数: 1

摘要

本文综述了通过[3+2]环加成在易获得的末端炔和磺酰叠氮之间直接合成具有重要生物意义的1-磺酰- 1,2,3 -三唑的方法。这篇评论分为两个主要部分。第一部分专门讨论1-(n -磺酰基)-4取代1,2,3-三唑的合成，而第二部分将讨论1-(n -磺酰基)-5取代1,2,3-三唑衍生物的制备。图形抽象

本文章由计算机程序翻译，如有差异，请以英文原文为准。

查看原文本刊更多论文

The synthesis of biologically active 1-sulfonyl-1, 2, 3-triazoles from sulfonyl azides and alkynes: a focus review

In this review, we spotlight the methods for the direct synthesis of synthetically and biologically important 1-sulfonyl-1, 2, 3-triazoles via [3+2] cycloaddition between easily available terminal alkynes and sulfonyl azides. The review is divided into two major sections. The first section focuses exclusively on the synthesis of 1-(N-sulfonyl)-4-substituted 1,2,3-triazoles, while the second section will discuss preparation of 1-(N-sulfonyl)-5-substituted 1,2,3-triazole derivatives.

求助全文

通过发布文献求助，成功后即可免费获取论文全文。去求助

来源期刊

Journal of Sulfur Chemistry CHEMISTRY, MULTIDISCIPLINARY-

CiteScore

4.10

自引率

9.10%

发文量

审稿时长

6-12 weeks

期刊介绍： The Journal of Sulfur Chemistry is an international journal for the dissemination of scientific results in the rapidly expanding realm of sulfur chemistry. The journal publishes high quality reviews, full papers and communications in the following areas: organic and inorganic chemistry, industrial chemistry, materials and polymer chemistry, biological chemistry and interdisciplinary studies directly related to sulfur science. Papers outlining theoretical, physical, mechanistic or synthetic studies pertaining to sulfur chemistry are welcome. Hence the target audience is made up of academic and industrial chemists with peripheral or focused interests in sulfur chemistry. Manuscripts that truly define the aims of the journal include, but are not limited to, those that offer: a) innovative use of sulfur reagents; b) new synthetic approaches to sulfur-containing biomolecules, materials or organic and organometallic compounds; c) theoretical and physical studies that facilitate the understanding of sulfur structure, bonding or reactivity; d) catalytic, selective, synthetically useful or noteworthy transformations of sulfur containing molecules; e) industrial applications of sulfur chemistry; f) unique sulfur atom or molecule involvement in interfacial phenomena; g) descriptions of solid phase or combinatorial methods involving sulfur containing substrates. Submissions pertaining to related atoms such as selenium and tellurium are also welcome. Articles offering routine heterocycle formation through established reactions of sulfur containing substrates are outside the scope of the journal.