Abdelrahman Y. Sherif*, and , Mohamed Abbas Ibrahim,
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In vitro dissolution was conducted to explore the influence of the formulation type on the dissolution profile of candesartan cilexetil (CC). The selected optimum L-SNEDDS formulation consisted of Tween-80:Imwitor-308:propylene glycol (2:1:1). The IL-SNEDDS formulation containing 7.5% w/w Pluronic-F-68 was selected as the optimum formulation with a liquefying temperature (34 °C) and liquefying time (75 s). Furthermore, physicochemical characterization revealed that candesartan cilexetil was present in the amorphous state within the prepared S-SNEDDS and IL-SNEDDS formulations, with no indication of a chemical interaction. In contrast to S-SNEDDS, IL-SNEDDS was able to enhance the dissolution of candesartan cilexetil with no sign of drug trapping. The present study presents a new approach that can overcome the limitations of traditional solid SNEDDS and enhance the application of SNEDDS as a pharmaceutical dosage form.</p>","PeriodicalId":22,"journal":{"name":"ACS Omega","volume":"10 37","pages":"43089–43100"},"PeriodicalIF":4.3000,"publicationDate":"2025-09-11","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"https://pubs.acs.org/doi/pdf/10.1021/acsomega.5c06315","citationCount":"0","resultStr":"{\"title\":\"Pluronic F-68 Triblock Copolymer Architecture for a Next-Generation Self-Nanoemulsifying System: Overcoming Drug Trapping and Dosage Challenges of Candesartan Cilexetil\",\"authors\":\"Abdelrahman Y. Sherif*, and , Mohamed Abbas Ibrahim, \",\"doi\":\"10.1021/acsomega.5c06315\",\"DOIUrl\":null,\"url\":null,\"abstract\":\"<p >Solidification of liquid self-nanoemulsifying drug delivery systems (L-SNEDDS) is commonly used to avoid formulation leakage during storage. However, traditional solidification using the adsorption method has limitations, including the trapping of drugs within adsorbent pores and the high total dosage required. Pluronic F-68, a triblock copolymer, was utilized to prepare a polymeric SNEDDS with an in situ liquefying property (IL-SNEDDS) using candesartan cilexetil as a model drug. Drug solubility was examined to choose the optimum L-SNEDDS formulation. Afterward, S-SNEDDS and IL-SNEDDS were prepared and subjected to physicochemical characterization. In vitro dissolution was conducted to explore the influence of the formulation type on the dissolution profile of candesartan cilexetil (CC). The selected optimum L-SNEDDS formulation consisted of Tween-80:Imwitor-308:propylene glycol (2:1:1). The IL-SNEDDS formulation containing 7.5% w/w Pluronic-F-68 was selected as the optimum formulation with a liquefying temperature (34 °C) and liquefying time (75 s). Furthermore, physicochemical characterization revealed that candesartan cilexetil was present in the amorphous state within the prepared S-SNEDDS and IL-SNEDDS formulations, with no indication of a chemical interaction. In contrast to S-SNEDDS, IL-SNEDDS was able to enhance the dissolution of candesartan cilexetil with no sign of drug trapping. 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Pluronic F-68 Triblock Copolymer Architecture for a Next-Generation Self-Nanoemulsifying System: Overcoming Drug Trapping and Dosage Challenges of Candesartan Cilexetil
Solidification of liquid self-nanoemulsifying drug delivery systems (L-SNEDDS) is commonly used to avoid formulation leakage during storage. However, traditional solidification using the adsorption method has limitations, including the trapping of drugs within adsorbent pores and the high total dosage required. Pluronic F-68, a triblock copolymer, was utilized to prepare a polymeric SNEDDS with an in situ liquefying property (IL-SNEDDS) using candesartan cilexetil as a model drug. Drug solubility was examined to choose the optimum L-SNEDDS formulation. Afterward, S-SNEDDS and IL-SNEDDS were prepared and subjected to physicochemical characterization. In vitro dissolution was conducted to explore the influence of the formulation type on the dissolution profile of candesartan cilexetil (CC). The selected optimum L-SNEDDS formulation consisted of Tween-80:Imwitor-308:propylene glycol (2:1:1). The IL-SNEDDS formulation containing 7.5% w/w Pluronic-F-68 was selected as the optimum formulation with a liquefying temperature (34 °C) and liquefying time (75 s). Furthermore, physicochemical characterization revealed that candesartan cilexetil was present in the amorphous state within the prepared S-SNEDDS and IL-SNEDDS formulations, with no indication of a chemical interaction. In contrast to S-SNEDDS, IL-SNEDDS was able to enhance the dissolution of candesartan cilexetil with no sign of drug trapping. The present study presents a new approach that can overcome the limitations of traditional solid SNEDDS and enhance the application of SNEDDS as a pharmaceutical dosage form.
ACS OmegaChemical Engineering-General Chemical Engineering
CiteScore
6.60
自引率
4.90%
发文量
3945
审稿时长
2.4 months
期刊介绍:
ACS Omega is an open-access global publication for scientific articles that describe new findings in chemistry and interfacing areas of science, without any perceived evaluation of immediate impact.