Chenghao Tang (Conceptualization Funding acquisition Writing – original draft Writing – review & editing) , Liang Chen (Data curation) , Qian Wang (Investigation) , Xiaoli Huang (Investigation) , Lanlan Wang (Data curation) , Wenting Yang (Validation) , Yue Zhou (Investigation) , Pei Li (Writing – original draft) , Xiang Wang (Writing – original draft)
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引用次数: 0
Abstract
A series of novel indole C2 derivatives containing 1,3,4-oxadiazole thioether moiety were designed and synthesized via natural compound indole-2-carboxylic acid as start material, and their biological activities were tested for Pseudomonas syringae pv actinidiae (Psa), Xanthomonas axonopodis pv citri (Xac), and Xanthomonas oryzae pv oryzae (Xoo). Bioassay findings revealed that a subset of the target compounds demonstrated robust antibacterial activities against Psa, Xoo and Xac at concentrations of both 100 and 50 μg/mL. Ongoing research is focused on exploring their bioactive applications, aiming to identify novel indole C2 derivatives and investigate their broad applicability.
期刊介绍:
Phosphorus, Sulfur, and Silicon and the Related Elements is a monthly publication intended to disseminate current trends and novel methods to those working in the broad and interdisciplinary field of heteroatom chemistry.