Elizaveta Karchuganova, Sofiia Martynova, Stanislav Kalinin, A. Angeli, Dmitry Dar'in, Daniella Vullo, C. Supuran, O. Bakulina
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Direct assembly of N-sulfamoyl lactam scaffolds bearing a zinc-binding group for inhibiting metalloenzymes based on desymmetrization of sulfamide and the Castagnoli-Cushman reaction