Samir, MESSAOUDI, Sokna , Bazzi, Ameni , Hadj Mohamed, Dmytro , Ryzhakov, Juba , Ghouilem, Mehdi A. , Beniddir, Vincent , Gandon
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引用次数: 0
Abstract
Here we report a macrocyclization route towards the
synthesis of glycophane peptides by a selective C-H arylation of the anomeric bond. This approach demonstrates the power of Pd-catalysis
C-H activation to access unfamiliar cyclic peptides