Preliminary screening of potential analgesics among cyanothioacetamide derivatives

E. Bibik, I. S. Oleĭnik, A. Saul, B. S. Krivokolysko, K. Frolov, V. Dotsenko, S. Krivokolysko
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Abstract

The aim of the research: to study the ability of cyanothioacetamide derivatives synthesized by us on the basis of the research laboratory “Khimeks”, Lugansk State University named after Volodymyr Dahl [1], which have low acute oral toxicity in experiments in vivo [2], to bind to potential biological targets.
氰硫乙酰胺衍生物潜在镇痛药的初步筛选
研究目的:研究我们在卢甘斯克国立大学“Khimeks”研究实验室的基础上合成的以Volodymyr Dahl命名的氰硫乙酰胺衍生物[1],该衍生物在体内实验中具有较低的急性口服毒性[2],与潜在的生物靶点结合的能力。
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