A. Klippel, Rui Wang, L. Puca, Andrew L. Faber, W. Shen, S. Bhagwat, Kannan R. Karukurichi, Feiyu Zhang, C. Pérez, Ramón Rama, Ana Ramos, Yi Zheng, Z. Bonday, James Thomas, H. Brooks, Lisa J. Kindler, Sarah M. Bogner, Parisa Zolfaghari, M. Ii, S. Callies, B. Mattioni, L. LeBrun, J. Durbin, E. Anderson, Chris Mayne, E. Kesicki, Gabrielle R. Kolakowski, S. Andrews, B. Brandhuber
{"title":"Abstract P142: Preclinical characterization of LOX-22783, a highly potent, mutant-selective and brain-penetrant allosteric PI3Kα H1047R inhibitor","authors":"A. Klippel, Rui Wang, L. Puca, Andrew L. Faber, W. Shen, S. Bhagwat, Kannan R. Karukurichi, Feiyu Zhang, C. Pérez, Ramón Rama, Ana Ramos, Yi Zheng, Z. Bonday, James Thomas, H. Brooks, Lisa J. Kindler, Sarah M. Bogner, Parisa Zolfaghari, M. Ii, S. Callies, B. Mattioni, L. LeBrun, J. Durbin, E. Anderson, Chris Mayne, E. Kesicki, Gabrielle R. Kolakowski, S. Andrews, B. Brandhuber","doi":"10.1158/1535-7163.targ-21-p142","DOIUrl":null,"url":null,"abstract":"","PeriodicalId":20348,"journal":{"name":"Poster Presentations - Proffered Abstracts","volume":"14 1","pages":""},"PeriodicalIF":0.0000,"publicationDate":"2021-12-01","publicationTypes":"Journal Article","fieldsOfStudy":null,"isOpenAccess":false,"openAccessPdf":"","citationCount":"2","resultStr":null,"platform":"Semanticscholar","paperid":null,"PeriodicalName":"Poster Presentations - Proffered Abstracts","FirstCategoryId":"1085","ListUrlMain":"https://doi.org/10.1158/1535-7163.targ-21-p142","RegionNum":0,"RegionCategory":null,"ArticlePicture":[],"TitleCN":null,"AbstractTextCN":null,"PMCID":null,"EPubDate":"","PubModel":"","JCR":"","JCRName":"","Score":null,"Total":0}