Patrycja Ledwoń, Michał Jewginski, Claudia Bello, Francesca Nuti, Paolo Rovero, Rafal Latajka, Anna Maria Papini
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引用次数: 0
Abstract
The Front Cover shows a set of Safirinium-dye derivatives used for the facile preparation of peptide conjugates as potential elastase inhibitors, by exploiting a lysine side chain as an effective linker between the dye and the peptide. With an optimized peptide sequence forming the core and triazolium derivatives acting as particular caps, we can create molecular tools capable of tuning the activity of a selected enzyme. Details of this approach are reported in the Research Article by R. Latajka, A. M. Papini and co-workers (DOI: 10.1002/ejoc.202400399). Structure taken from PDB ID: 1QR3.
期刊介绍：
The European Journal of Organic Chemistry (2019 ISI Impact Factor 2.889) publishes Full Papers, Communications, and Minireviews from the entire spectrum of synthetic organic, bioorganic and physical-organic chemistry. It is published on behalf of Chemistry Europe, an association of 16 European chemical societies.
The following journals have been merged to form two leading journals, the European Journal of Organic Chemistry and the European Journal of Inorganic Chemistry:
Liebigs Annalen
Bulletin des Sociétés Chimiques Belges
Bulletin de la Société Chimique de France
Gazzetta Chimica Italiana
Recueil des Travaux Chimiques des Pays-Bas
Anales de Química
Chimika Chronika
Revista Portuguesa de Química
ACH—Models in Chemistry
Polish Journal of Chemistry.
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